SCHEMBL9364015

SCHEMBL9364015

CCCOC(=O)OC1=C(C)N(C)C(C)=C(OC(=O)OC)C1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
HTT P42858 1/20 0.41
KDM4E B2RXH2 3/20 0.39
GAA P10253 2/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
NPSR1 Q6W5P4 3/20 0.37
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
BCHE P06276 2/20 0.36
ACHE P22303 2/20 0.36
ATM Q13315 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
KDM1A O60341 1/20 0.34
RCOR1 Q9UKL0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9364248 0.92 HSP90AA1 (0.44) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL8984936 0.90 HSP90AA1 (0.46) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL9364528 0.88 NPSR1 (0.45) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL7428174 0.84 HSP90AA1 (0.43) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL9364254 0.84 HSP90AA1 (0.40) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL9363808 0.84 HSP90AA1 (0.42) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL9364256 0.82 KDM4E (0.44) HSP90AA1HSP90AB1KDM4EGAAALDH1A1
SCHEMBL9364532 0.82 POLB (0.43) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL9364057 0.82 HSP90AA1 (0.41) HSP90AA1HSP90AB1HTTKDM4EGAA
SCHEMBL9363819 0.81 KDM4E (0.42) KDM4EGAAALDH1A1POLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP claimed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP claimed
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP disclosed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP disclosed