SCHEMBL9364392

SCHEMBL9364392

CC(C#N)c1ccc(-n2ccnc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
ENPP2 Q13822 1/20 0.50
MKNK1 Q9BUB5 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
NOTUM Q6P988 1/20 0.50
CYP3A4 P08684 3/20 0.49
BAZ2B Q9UIF8 1/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP19A1 P11511 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
HTR2A P28223 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL801703 0.81 NOTUM (0.63) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL6892003 0.78 NOTUM (0.59) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL8047855 0.78 LMNA (0.55) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL8278915 0.78 LMNA (0.59) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL6895118 0.78 ENPP2 (0.59) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL4876009 0.78 LMNA (0.44) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL2532397 0.76 LMNA (0.78) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL10311213 0.75 CYP3A4 (0.53) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL14438346 0.74 TDP1 (0.56) LMNAMAPTENPP2MKNK1MKNK2
SCHEMBL27513743 0.74 CYP3A4 (0.59) LMNAMAPTENPP2MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445698-B1 Thiocarbamoylacetonitrile compounds MITSUBISHI CHEM IND (JP) 1994-06-22 EP disclosed
US-5246958-A Thiocarbamoylacetonitriles MITSUBISHI KASEI CORPORATION (JP) 1993-09-21 US disclosed
EP-0445698-A1 Thiocarbamoylacetonitrile compounds MITSUBISHI KASEI CORPORATION (JP) 1991-09-11 EP disclosed
US-4226878-A ANTIINFLAMMATORY, HYPOTENSIVES, ANTIHISTAMINES KISSEI PHARMACEUTICAL CO., LTD. (JP) 1980-10-07 US disclosed