SCHEMBL9364584

SCHEMBL9364584

N#Cc1cc2[nH]c(=O)c(=O)n(O)c2cc1C#N

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 4/20 0.41
GRIA2 P42262 4/20 0.41
GRIA3 P42263 4/20 0.41
GRIA4 P48058 4/20 0.41
CYP1A2 P05177 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
DAO P14920 3/20 0.38
MAOA P21397 3/20 0.36
MAOB P27338 3/20 0.36
GRIN2D O15399 3/20 0.35
GRIN3B O60391 3/20 0.35
GRIN1 Q05586 3/20 0.35
GRIN2A Q12879 3/20 0.35
GRIN2B Q13224 3/20 0.35
GRIN2C Q14957 3/20 0.35
GRIN3A Q8TCU5 3/20 0.35
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9365335 0.88 GRIA1 (0.45) GRIA1GRIA2GRIA3GRIA4CYP1A2
SCHEMBL9364720 0.84 L3MBTL1 (0.40) GRIA1GRIA2GRIA3GRIA4CYP1A2
SCHEMBL9091900 0.84 GRIA1 (0.40) GRIA1GRIA2GRIA3GRIA4KDM4E
SCHEMBL9365531 0.78 FASN (0.44) DAO
SCHEMBL9362677 0.74 KDM4E (0.40) MAOAMAOBKDM4E
SCHEMBL9364622 0.74 GRIN2D (0.58) GRIA1GRIA2GRIA3GRIA4DAO
SCHEMBL4704409 0.74 GRIA1 (0.64) GRIA1GRIA2GRIA3GRIA4CYP1A2
SCHEMBL9971326 0.73 GRIA1 (0.63) GRIA1GRIA2GRIA3GRIA4CYP1A2
SCHEMBL9364640 0.72 DAO (0.39) GRIA1GRIA2GRIA3GRIA4DAO
SCHEMBL9368432 0.70 GRIN2D (0.56) DAOGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377112-B1 Quinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-08-24 EP disclosed
US-5061706-A 2,3-QUINOXALINEDIONES FOR USE AS NEUROLEPTICS NOVO NORDISK A/S (DK) 1991-10-29 US disclosed
EP-0377112-A1 Quinoxaline compounds and their preparation and use NOVO NORDISK A/S (DK) 1990-07-11 EP disclosed