Pha-665752

Pha-665752

SCHEMBL93655

Cc1[nH]c(/C=C2\C(=O)Nc3ccc(S(=O)(=O)Cc4c(Cl)cccc4Cl)cc32)c(C)c1C(=O)N1CCCC1CN1CCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 1.00
FGFR1 P11362 9/20 1.00
PDGFRB P09619 9/20 1.00
MET P08581 7/20 1.00
SRC P12931 6/20 1.00
LCK P06239 4/20 1.00
YES1 P07947 4/20 1.00
CDK2 P24941 2/20 1.00
PTK2B Q14289 2/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
KIT P10721 2/20 1.00
EGFR P00533 2/20 1.00
ALK Q9UM73 2/20 1.00
PLK4 O00444 1/20 1.00
RIOK3 O14730 1/20 1.00
CASK O14936 1/20 1.00
GAK O14976 1/20 1.00
DCLK1 O15075 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pha-665752 SCHEMBL29376386 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93656 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93657 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL140412 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93654 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL15639801 0.99 KDR (0.99) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL15639803 0.99 KDR (0.99) KDRFGFR1PDGFRBMETSRC
SCHEMBL23691031 0.97 KDR (0.94) KDRFGFR1PDGFRBMETSRC
SCHEMBL143795 0.96 KDR (0.93) KDRFGFR1PDGFRBMETSRC
SCHEMBL147331 0.95 KDR (0.91) KDRFGFR1PDGFRBMETSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2425830-A1 Synergistic drug combination for the treatment of cancer Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2012-03-07 EP claimed
CN-113164480-B Pharmaceutical composition for treating diffuse gastric cancer 学校法人金泽医科大学 2023-11-28 CN disclosed
CN-113164480-A Pharmaceutical composition for treating diffuse gastric cancer 学校法人金泽医科大学 2021-07-23 CN disclosed
CN-104762371-B Biomarkers for predicting or monitoring the efficacy of c-Met inhibitors 三星电子株式会社 2021-03-09 CN disclosed
US-20210047618-A1 Improved Differentiation Method KONINKLIJKE NEDERLANDSE AKADEMIE VAN WETENSCHAPPEN (NL) 2021-02-18 US disclosed
US-20160058751-A1 COMPOSITION AND METHOD FOR TREATING CANCER CELLWORKS GROUP, INC. (US) 2016-03-03 US disclosed
US-20160058751-A1 COMPOSITION AND METHOD FOR TREATING CANCER CELLWORKS GROUP, INC. (US) 2016-03-03 US disclosed
WO-2014160729-A1 COMPOSITION AND METHOD FOR TREATING CANCER CELLWORKS RESEARCH INDIA PVT. LTD (IN) 2014-10-02 WO disclosed
WO-2012028334-A2 MARKER FOR SUNITINIB RESISTANCE FORMATION MAX-PLANCK-GESELLSCHAFT ZUR FÖRDERUNG DER FÖRDERUNG DER WISSENSCHAFTEN E.V. (DE) 2012-03-08 WO disclosed
EP-2425830-A1 Synergistic drug combination for the treatment of cancer Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2012-03-07 EP disclosed
EP-2426213-A1 Marker for sunitnib resistance formation Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2012-03-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160058751-A1 COMPOSITION AND METHOD FOR TREATING CANCER KRAS, NRAS, TP53 KDR 953/4885FGFR1 1911/4885PDGFRB 1100/4885
US-20210047618-A1 Improved Differentiation Method VIPR2, IAPP, PROX1 KDR 3019/4885FGFR1 2149/4885PDGFRB 1923/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.