Pha-665752

Pha-665752

SCHEMBL29376386

Cc1[nH]c(/C=C2\C(=O)Nc3ccc(S(=O)(=O)Cc4c(Cl)cccc4Cl)cc32)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 1.00
FGFR1 P11362 9/20 1.00
PDGFRB P09619 9/20 1.00
MET P08581 7/20 1.00
SRC P12931 6/20 1.00
LCK P06239 4/20 1.00
YES1 P07947 4/20 1.00
CDK2 P24941 2/20 1.00
PTK2B Q14289 2/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
KIT P10721 2/20 1.00
EGFR P00533 2/20 1.00
ALK Q9UM73 2/20 1.00
PLK4 O00444 1/20 1.00
RIOK3 O14730 1/20 1.00
CASK O14936 1/20 1.00
GAK O14976 1/20 1.00
DCLK1 O15075 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pha-665752 SCHEMBL93656 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93657 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93655 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL140412 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93654 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL15639801 0.99 KDR (0.99) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL15639803 0.99 KDR (0.99) KDRFGFR1PDGFRBMETSRC
SCHEMBL23691031 0.97 KDR (0.94) KDRFGFR1PDGFRBMETSRC
SCHEMBL143795 0.96 KDR (0.93) KDRFGFR1PDGFRBMETSRC
SCHEMBL147331 0.95 KDR (0.91) KDRFGFR1PDGFRBMETSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 483 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4640238-A1 THERAPEUTIC AGENT FOR PULMONARY DISEASE, HEPATIC DISEASE OR RENAL DISEASE, WHICH CONTAINS PGAM-CHK1 BINDING INHIBITOR Kyoto University (JP) 2025-10-29 EP claimed
EP-4633630-A1 TREATMENT OF CANCER RESISTANT TO EGFR TKI USING C-MET INHIBITOR Apollomics Inc. (US) 2025-10-22 EP claimed
EP-4615869-A1 COMBINATION THERAPY COMPRISING BISPECIFIC ANTIBODIES COMPRISING AN NRP1 BINDING DOMAIN Pinetree Therapeutics, Inc. (US) 2025-09-17 EP claimed
US-20250270651-A1 DETECTION OF MET AMPLIFICATION TO PREDICT RESPONSIVENESS OF CANCER TO DRUGS THE GENERAL HOSPITAL CORPORATION (US) 2025-08-28 US claimed
US-20250003952-A1 SENOLYTIC DRUG SCREENING METHOD AND SENOLYTIC DRUG KYOTO UNIVERSITY (JP) 2025-01-02 US claimed
US-20240398801-A1 TREATMENT OF LEUKEMIA BASED ON LEUKEMIA HIERARCHY IN A PATIENT UNIVERSITY HEALTH NETWORK (CA) 2024-12-05 US claimed
EP-4423302-A2 NOVEL KINASE FUSIONS DETECTED BY LIQUID BIOPSY Foundation Medicine, Inc. (US) 2024-09-04 EP claimed
CN-118414439-A Novel kinase fusion by liquid biopsy 基金会医学公司 2024-07-30 CN claimed
EP-4400117-A1 SENOLYTIC DRUG SCREENING METHOD AND SENOLYTIC DRUG Kyoto University (JP) 2024-07-17 EP claimed
US-20240218453-A1 DIAGNOSTIC AND TREATMENT OF CANCER USING C-MET INHIBITOR APOLLOMICS INC. 2024-07-04 US claimed
WO-2023050018-A1 TREATMENT OF LEUKEMIA BASED ON LEUKEMIA HIERARCHY IN A PATIENT UNIVERSITY HEALTH NETWORK (CA) 2023-04-06 WO claimed
WO-2023038027-A1 SENOLYTIC DRUG SCREENING METHOD AND SENOLYTIC DRUG 国立大学法人京都大学 2023-03-16 WO claimed
US-11583544-B2 Remote loading of sparingly water-soluble drugs into lipid vesicles CELATOR PHARMACEUTICALS, INC. (US) 2023-02-21 US claimed
US-20220412957-A1 METHODS OF TREATING CANCER PATIENTS WITH RAS NODE OR RTK TARGETED THERAPEUTIC AGENTS OXFORD FINANCE LLC, AS COLLATERAL AGENT 2022-12-29 US claimed
WO-2022226168-A1 DIAGNOSTIC AND TREATMENT OF CANCER USING C-MET INHIBITOR APOLLOMICS INC. (US) 2022-10-27 WO claimed
EP-4073516-A1 METHODS OF TREATING CANCER PATIENTS WITH RAS NODE OR RTK TARGETED THERAPEUTIC AGENTS Celcuity Inc. (US) 2022-10-19 EP claimed
US-20220252603-A1 METHOD FOR TREATING CANCER PATIENTS USING C-MET INHIBITOR APOLLOMICS INC. (HANGZHOU) (CN) 2022-08-11 US claimed
CN-114599978-A Methods of treating cancer patients using C-MET inhibitors 浙江冠科美博生物科技有限公司 2022-06-07 CN claimed
EP-3980783-A1 METHOD FOR TREATING CANCER PATIENTS USING C-MET INHIBITOR Apollomics Inc. (Hangzhou) (CN) 2022-04-13 EP claimed
EP-3964206-A1 COMPOUNDS FOR THE TREATMENT OF COVID-19 Dompe' Farmaceutici S.P.A. (IT) 2022-03-09 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240218453-A1 DIAGNOSTIC AND TREATMENT OF CANCER USING C-MET INHIBITOR MET, METTL16, HGF KDR 516/4885FGFR1 150/4885PDGFRB 94/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.