Pha-665752

Pha-665752

SCHEMBL93654

Cc1[nH]c(/C=C2\C(=O)Nc3ccc(S(=O)(=O)Cc4c(Cl)cccc4Cl)cc32)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 1.00
FGFR1 P11362 9/20 1.00
PDGFRB P09619 9/20 1.00
MET P08581 7/20 1.00
SRC P12931 6/20 1.00
LCK P06239 4/20 1.00
YES1 P07947 4/20 1.00
CDK2 P24941 2/20 1.00
PTK2B Q14289 2/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
KIT P10721 2/20 1.00
EGFR P00533 2/20 1.00
ALK Q9UM73 2/20 1.00
PLK4 O00444 1/20 1.00
RIOK3 O14730 1/20 1.00
CASK O14936 1/20 1.00
GAK O14976 1/20 1.00
DCLK1 O15075 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pha-665752 SCHEMBL29376386 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93656 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93657 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL93655 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL140412 1.00 KDR (1.00) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL15639801 0.99 KDR (0.99) KDRFGFR1PDGFRBMETSRC
Pha-665752 SCHEMBL15639803 0.99 KDR (0.99) KDRFGFR1PDGFRBMETSRC
SCHEMBL23691031 0.97 KDR (0.94) KDRFGFR1PDGFRBMETSRC
SCHEMBL143795 0.96 KDR (0.93) KDRFGFR1PDGFRBMETSRC
SCHEMBL147331 0.95 KDR (0.91) KDRFGFR1PDGFRBMETSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 193 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8729043-B2 Anti-Met monoclonal antibody, fragments and vectors thereof, for the treatment of tumors and corresponding products METHERESIS TRANSLATIONAL RESEARCH S.A. (CH) 2014-05-20 US claimed
EP-2425830-A1 Synergistic drug combination for the treatment of cancer Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2012-03-07 EP claimed
EP-1981981-B1 ANTI-MET MONOCLONAL ANTIBODY, FRAGMENTS AND VECTORS THEREOF, FOR THE TREATMENT OF TUMORS AND CORRESPONDING PRODUCTS METHERESIS TRANSLATIONAL RES SA (CH) 2011-06-29 EP claimed
US-20090285807-A1 Anti-Met Monoclonal Antibody, Fragments and Vectors Thereof, for the Treatment of Tumors and Corresponding Products Pierre Fabre Médicament (FR) 2009-11-19 US claimed
US-6599902-B2 For treating or preventing a protein kinase related disorder SUGEN, INC. 2003-07-29 US claimed
US-20030125370-A1 5-ARALKYSUFONYL-3-(PYRROL-2-YLMETHYLIDENE)-2-INDOLINONE DERIVATIVES AS KINASE INHIBITORS SUGEN, INC. 2003-07-03 US claimed
WO-2002096361-A2 5-ARALKYLSULFONYL-3- (PYRROL-2-YLMETHYLIDENE)-2-INDOLINONE DERIVATIVES AS KINASE INHIBITORS SUGEN, INC. (US) 2002-12-05 WO claimed
US-12570625-B2 3-(5-hydroxy-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2026-03-10 US disclosed
EP-4541381-B1 STABLE, CONCENTRATED RADIONUCLIDE COMPLEX SOLUTIONS ADVANCED ACCELERATOR APPLICATIONS S A (FR) 2026-02-04 EP disclosed
EP-4545100-B1 STABLE, CONCENTRATED RADIONUCLIDE COMPLEX SOLUTIONS ADVANCED ACCELERATOR APPLICATIONS S A (FR) 2025-12-10 EP disclosed
EP-4545101-B1 STABLE, CONCENTRATED RADIONUCLIDE COMPLEX SOLUTIONS ADVANCED ACCELERATOR APPLICATIONS S A (FR) 2025-12-10 EP disclosed
EP-4541380-B1 STABLE, CONCENTRATED RADIONUCLIDE COMPLEX SOLUTIONS ADVANCED ACCELERATOR APPLICATIONS S A (FR) 2025-12-10 EP disclosed
US-12479817-B2 Substituted 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2025-11-25 US disclosed
WO-2007009613-A1 METHOD FOR MEASURING TYROSINE KINASE PHOSPHORYLATION MERCK PATENT GMBH (DE) 2007-01-25 WO disclosed
US-20060246492-A1 Method for predicting responsiveness to drugs THE GENERAL HOSPITAL CORPORATION (US) 2006-11-02 US disclosed
US-20060035907-A1 Methods of treating abnormal cell growth using c-MET and m-TOR inhibitors CHRISTENSEN JAMES G 2006-02-16 US disclosed
US-20050282733-A1 Differentiation modulating agents and uses therefor VERVA PHARMACEUTICALS PTY LTD (AU) 2005-12-22 US disclosed
WO-2005082411-A1 METHOD OF TREATING ABNORMAL CELL GROWTH USING C-MET AND-TOR INHIBITORS SUGEN, INC. (US) 2005-09-09 WO disclosed
US-6599902-B2 For treating or preventing a protein kinase related disorder SUGEN, INC. 2003-07-29 US disclosed
US-20030125370-A1 5-ARALKYSUFONYL-3-(PYRROL-2-YLMETHYLIDENE)-2-INDOLINONE DERIVATIVES AS KINASE INHIBITORS SUGEN, INC. 2003-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035907-A1 Methods of treating abnormal cell growth using c-MET and m-TOR inhibitors MET, MTOR, MYC KDR 252/4885FGFR1 68/4885PDGFRB 560/4885
US-12479817-B2 Substituted 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof XDH, RXFP3, NPY2R KDR 2878/4885FGFR1 2771/4885PDGFRB 4228/4885
US-12570625-B2 3-(5-hydroxy-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof IKZF1, IKZF2, BCL6 KDR 3515/4885FGFR1 2064/4885PDGFRB 4669/4885
US-20050282733-A1 Differentiation modulating agents and uses therefor FGF1, FABP4, FGF2 KDR 1077/4885FGFR1 5/4885PDGFRB 467/4885
US-20030125370-A1 5-ARALKYSUFONYL-3-(PYRROL-2-YLMETHYLIDENE)-2-INDOLINONE DERIVATIVES AS KINASE INHIBITORS DMPK, ADK, MAP3K20 KDR 398/4885FGFR1 637/4885PDGFRB 348/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.