SCHEMBL936563

SCHEMBL936563

OCC1CCc2ccccc2O1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.55
HTR1A P08908 9/20 0.52
SIGMAR1 Q99720 2/20 0.52
ADRA2A P08913 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
HTR1D P28221 6/20 0.49
DRD2 P14416 2/20 0.43
DRD4 P21917 2/20 0.43
DRD3 P35462 2/20 0.43
DRD1 P21728 1/20 0.43
DRD5 P21918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5722925 1.00 CA2 (0.55) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL7346709 1.00 CA2 (0.55) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL30711484 1.00 CA2 (0.55) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL7145238 0.89 CA2 (0.46) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL4823736 0.89 CA2 (0.60) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL4823732 0.89 CA2 (0.60) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL8935393 0.86 CA2 (0.52) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL8935402 0.86 CA2 (0.52) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL10645332 0.86 CA2 (0.52) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL4936349 0.83 CA2 (0.56) CA2HTR1ASIGMAR1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 255 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108299364-B A kind of synthetic method of 2- methylol chromanone 常州大学 2019-07-09 CN claimed
US-20050014818-A1 Process for producing optically active chroman derivative and intermediate KANEKA CORPORATION (JP) 2005-01-20 US claimed
CN-1564818-A Stereoselective synthesis method of 2-hydroxymethyl-chroman WYETH CORP (US) 2005-01-12 CN claimed
EP-1445324-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE CHROMAN DERIVATIVE AND INTERMEDIATE KANEKA CORPORATION (JP) 2004-08-11 EP claimed
EP-1432695-A1 A PROCESS FOR THE STEREOSELECTIVE SYNTHESIS OF 2-HYDROXYMETHYL-CHROMANS Wyeth (US) 2004-06-30 EP claimed
US-6700001-B2 USEFUL AS INTERMEDIATES TO DRUGS INCLUDING THOSE TO TREAT CENTRAL NERVOUS SYSTEM DISORDERS; STEREOSPECIFIC CYCLIZATION OF AN OPTICALLY ACTIVE PHENOL COMPOUND WYETH 2004-03-02 US claimed
US-20030105342-A1 Process for stereoselective synthesis of 2-hydroxymethyl chromans WYETH 2003-06-05 US claimed
WO-2003031429-A1 A PROCESS FOR THE STEREOSELECTIVE SYNTHESIS OF 2-HYDROXYMETHYL-CHROMANS WYETH (US) 2003-04-17 WO claimed
EP-0801564-B1 USE OF NEBIVOLOL AS AN ANTI-ATHEROGENIC JANSSEN PHARMACEUTICA NV (BE) 2002-03-27 EP claimed
EP-0801564-A1 USE OF NEBIVOLOL AS AN ANTI-ATHEROGENIC JANSSEN PHARMACEUTICA N.V. (BE) 1997-10-22 EP claimed
WO-1996019987-A1 USE OF NEBIVOLOL AS AN ANTI-ATHEROGENIC JANSSEN PHARMACEUTICA N.V. (BE) 1996-07-04 WO claimed
EP-0448254-B1 Process and intermediates for 2R-benzyl-chroman-6-carbaldehyde PFIZER (US) 1995-01-18 EP claimed
EP-0448254-A2 Process and intermediates for 2R-benzyl-chroman-6-carbaldehyde PFIZER INC. (US) 1991-09-25 EP claimed
US-4515975-A Chroman derivatives and their preparation BASF AKTIENGESELLSCHAFT (DE) 1985-05-07 US claimed
EP-0052731-B1 CHROMAN DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF Aktiengesellschaft (DE) 1985-04-17 EP claimed
EP-4134364-B1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RES INC (US) 2025-07-30 EP disclosed
US-20240182490-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2024-06-06 US disclosed
US-4374258-A PHOTOSTABILITY; HEAT AND OXIDATION RESISTANCE; ADDITION POLYMERS BASF AKTIENGESELLSCHAFT (DE) 1983-02-15 US disclosed
EP-0057425-A1 Chromane derivatives BASF Aktiengesellschaft (DE) 1982-08-11 EP disclosed
EP-0052731-A1 Chroman derivatives and method for their preparation BASF Aktiengesellschaft (DE) 1982-06-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240182490-A1 BROMODOMAIN INHIBITORS BRD3, EP300, BRPF3 CA2 3892/4885HTR1A 4461/4885SIGMAR1 4496/4885
US-20050014818-A1 Process for producing optically active chroman derivative and intermediate CYP8B1, CYP3A43, HPD CA2 825/4885HTR1A 739/4885SIGMAR1 1763/4885
US-20030105342-A1 Process for stereoselective synthesis of 2-hydroxymethyl chromans CYP2S1, CYP1B1, CYP1A2 CA2 2495/4885HTR1A 57/4885SIGMAR1 3078/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.