SCHEMBL9366390

SCHEMBL9366390

CCOc1ccc2nc(Cl)c(S(N)(=O)=O)n2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
TNF P01375 1/20 0.36
PTGS2 P35354 4/20 0.35
PTGS1 P23219 3/20 0.35
CA1 P00915 5/20 0.35
CA2 P00918 5/20 0.35
CA9 Q16790 5/20 0.35
CA12 O43570 3/20 0.35
CA7 P43166 2/20 0.35
CA14 Q9ULX7 2/20 0.33
MKNK1 Q9BUB5 2/20 0.33
PDE10A Q9Y233 3/20 0.32
KDM4E B2RXH2 2/20 0.32
LMNA P02545 1/20 0.32
CA3 P07451 1/20 0.32
PKM P14618 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9362850 0.90 CA12 (0.38) HTTAKT1AKT2TNFPTGS2
SCHEMBL3342309 0.85 HTT (0.40) HTTAKT1AKT2CA1CA2
SCHEMBL9367773 0.85 DYRK1A (0.38) HTTAKT1AKT2TNFPTGS2
SCHEMBL3342795 0.84 AKT1 (0.40) HTTAKT1AKT2PTGS2CA1
SCHEMBL3343151 0.82 AKT1 (0.39) HTTAKT1AKT2CA1CA2
SCHEMBL3346028 0.82 CHRNA7 (0.35) TNFPTGS2
SCHEMBL3343016 0.81 PDE10A (0.40) HTTAKT1AKT2PTGS2PTGS1
SCHEMBL2065760 0.80 TNF (0.35) AKT1AKT2TNFCA1CA2
SCHEMBL2065746 0.77 PDE10A (0.37) TNFCA1CA2CA12CA7
SCHEMBL3157242 0.77 TNF (0.54) AKT1AKT2TNFMKNK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0305939-B1 Process of producing sulfonylurea derivatives TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1994-11-02 EP disclosed
US-4994571-A Reacting heterocycle-containing sulfonamide compound with carbonyl compound TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-02-19 US disclosed
EP-0305939-A1 Process of producing sulfonylurea derivatives Takeda Chemical Industries, Ltd. (JP) 1989-03-08 EP disclosed