SCHEMBL9368018

SCHEMBL9368018

COc1ccc(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)cc1OC

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 10/20 0.72
HTR2C P28335 5/20 0.72
HTR7 P34969 4/20 0.72
HTR6 P50406 3/20 0.72
MAPT P10636 2/20 0.68
HTT P42858 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
GRM2 Q14416 3/20 0.63
KMT2A Q03164 2/20 0.59
DRD2 P14416 2/20 0.56
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 1/20 0.56
MAPK1 P28482 1/20 0.56
CYP2D6 P10635 2/20 0.55
KCNH2 Q12809 1/20 0.55
KDM4E B2RXH2 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C19 P33261 1/20 0.55
HTR1A P08908 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9362999 0.99 HTR2A (0.71) HTR2AHTR2CHTR7HTR6MAPT
SCHEMBL10508915 0.89 MAPT (0.59) HTR2AHTR2CHTR7HTR6MAPT
SCHEMBL9444495 0.84 KCNH2 (0.58) HTR2AHTR2CHTR7HTR6MAPT
SCHEMBL27334030 0.84 SIGMAR1 (0.56) HTR2AGRM2KMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL9444430 0.83 KCNH2 (0.59) HTR2AHTR2CHTR7HTR6MAPT
SCHEMBL9500292 0.82 ALDH1A1 (0.69) HTR2AHTR2CHTR7HTR6MAPT
SCHEMBL10709567 0.82 HTR2A (0.53) HTR2AHTR2CHTR7HTR6MAPT
SCHEMBL1583307 0.82 HTR2A (0.88) HTR2AHTR2CHTR7HTR6GRM2
SCHEMBL9363920 0.81 HTR2A (0.55) HTR2AHTR2CHTR7HTR6MAPT
SCHEMBL1582719 0.81 KCNH2 (0.83) HTR2AHTR2CHTR7HTR6CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360275-B1 Imidazole antiarrhythmics MERRELL DOW PHARMA (US) 1994-01-12 EP disclosed
EP-0360275-A2 Imidazole antiarrhythmics MERRELL DOW PHARMACEUTICALS INC. (US) 1990-03-28 EP disclosed
US-4868194-A Imidazole antiarrhythmics MERRELL DOW PHARMACEUTICALS INC. (US) 1989-09-19 US disclosed