SCHEMBL9369986

SCHEMBL9369986

Fc1ccccc1Cn1nnc2c(NC3CC3)nccc21

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.53
ALDH1A1 P00352 5/20 0.45
PKM P14618 2/20 0.44
POLB P06746 1/20 0.44
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9370128 0.87 GRM2 (0.45) GRM2ALDH1A1ADORA3ADORA2AADORA2B
SCHEMBL9373426 0.84 GRM2 (0.56) GRM2ALDH1A1PKMPOLBADORA3
Hydrochloric Acid SCHEMBL9375536 0.83 GRM2 (0.55) GRM2ALDH1A1PKMPOLBADORA3
SCHEMBL9369141 0.82 GRM2 (0.54) GRM2ALDH1A1PKMPOLBADORA3
SCHEMBL9368312 0.75 GRM2 (0.56) GRM2ALDH1A1PKMPOLBADORA3
SCHEMBL9369054 0.71 GRM2 (0.42) GRM2ALDH1A1POLBADORA3ADORA2A
SCHEMBL9370038 0.71 ADORA3 (0.42) GRM2ALDH1A1ADORA3ADORA2AADORA2B
Hydrochloric Acid SCHEMBL9368834 0.70 GRM2 (0.41) GRM2ALDH1A1POLBADORA3ADORA2A
SCHEMBL9735164 0.69 ALDH1A1 (0.44) GRM2ALDH1A1PKMPOLBADORA3
Hydrochloric Acid SCHEMBL9735017 0.68 ALDH1A1 (0.43) GRM2ALDH1A1PKMPOLBADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0399653-B1 Anticonvulsant triazolo[4,5-c]pyridine derivatives WELLCOME FOUND (GB) 1994-10-19 EP claimed
US-5240937-A Treatment of epilepsy BURROUGHS WELLCOME CO. (US) 1993-08-31 US claimed
EP-0399653-A1 Anticonvulsant triazolo[4,5-c]pyridine derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1990-11-28 EP claimed
US-5240937-A Treatment of epilepsy BURROUGHS WELLCOME CO. (US) 1993-08-31 US disclosed
EP-0399653-A1 Anticonvulsant triazolo[4,5-c]pyridine derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1990-11-28 EP disclosed