SCHEMBL9374602

SCHEMBL9374602

CCCc1cc(C(=O)CBr)ccc1OC

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.50
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ALOX5 P09917 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRB2 P47870 1/20 0.44
HPGDS O60760 1/20 0.43
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
HMGCR P04035 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6343700 0.83 ALDH1A1 (0.65) ALDH1A1MEN1KMT2AMAPT
SCHEMBL3547262 0.83 CA12 (0.61) ALDH1A1MEN1KMT2AALOX5GABRA1
SCHEMBL9373198 0.82 THRA (0.52) CTNNB1WNT3A
SCHEMBL3543244 0.81 MAPT (0.55) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL20058880 0.81 MAPK1 (0.60) ALDH1A1MEN1KMT2AALOX5GABRA1
SCHEMBL29620831 0.80 TSHR (0.63) GSK3BALDH1A1MEN1KMT2ACTNNB1
SCHEMBL426444 0.80 TSHR (0.63) GSK3BALDH1A1MEN1KMT2ACTNNB1
SCHEMBL10955996 0.80 PDE4B (0.55) ALDH1A1MEN1KMT2ACTNNB1WNT3A
SCHEMBL4344454 0.80 HTT (0.48) GSK3BALDH1A1ALOX5MAPT
SCHEMBL9378829 0.78 ALDH1A1 (0.45) ALDH1A1MEN1KMT2AALOX5GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0607217-A1 PYRIDINOL DERIVATIVES AS MEDICAMENTS SMITHKLINE BEECHAM PLC (GB) 1994-07-27 EP disclosed
WO-1993007137-A1 PYRIDINOL DERIVATIVES AS MEDICAMENTS SMITHKLINE BEECHAM PLC (GB) 1993-04-15 WO disclosed