SCHEMBL9375237

SCHEMBL9375237

NC(=O)c1ccc2c(c1)CCC(=O)N2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.61
SMYD3 Q9H7B4 2/20 0.58
CRBN Q96SW2 5/20 0.54
HDAC3 O15379 2/20 0.50
HDAC4 P56524 2/20 0.50
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
HDAC9 Q9UKV0 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
NPC1 O15118 1/20 0.49
MAPK13 O15264 1/20 0.49
MAPK12 P53778 1/20 0.49
MAPK11 Q15759 1/20 0.49
MAPK14 Q16539 1/20 0.49
KIF11 P52732 1/20 0.48
CA9 Q16790 1/20 0.47
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9379920 0.88 CA9 (0.62) SIRT2SMYD3CRBNNPC1MAPK13
SCHEMBL3307683 0.88 KIF11 (0.61) SIRT2SMYD3CRBNHDAC3HDAC4
SCHEMBL27599042 0.87 CRBN (0.54) SIRT2SMYD3CRBNHDAC3HDAC4
SCHEMBL3190474 0.85 SMYD3 (0.57) SIRT2SMYD3HDAC3
SCHEMBL939611 0.85 SMYD3 (0.59) SMYD3CRBNHDAC3HDAC4HDAC1
SCHEMBL29567045 0.85 SMYD3 (0.57) SIRT2SMYD3HDAC3
SCHEMBL29995492 0.85 SMYD3 (0.59) SMYD3CRBNHDAC3HDAC4HDAC1
SCHEMBL3312591 0.84 TDP2 (0.60) SIRT2SMYD3CRBNNPC1KIF11
Hydrochloric Acid SCHEMBL28849276 0.83 SMYD3 (0.56) SIRT2SMYD3HDAC3
Succinimide SCHEMBL9294241 0.83 SMYD3 (0.58) SMYD3CRBNHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023122212-A2 SUBSTITUTED PHENYL ETHYNYL PYRIDINE CARBOXAMIDES AS POTENT INHIBITORS OF SARS VIRUS SOUTHERN RESEARCH INSTITUTE (US) 2023-06-29 WO disclosed
EP-0344634-B1 Bicyclic carboxamides, process for their preparation and medicaments containing them BOEHRINGER MANNHEIM GMBH (DE) 1994-03-30 EP disclosed
US-5019587-A Anticoagulants BOEHRINGER MANNHEIM GMBH (DE) 1991-05-28 US disclosed
EP-0344634-A1 Bicyclic carboxamides, process for their preparation and medicaments containing them Roche Diagnostics GmbH (DE) 1989-12-06 EP disclosed