SCHEMBL9375259

SCHEMBL9375259

CC1(C)CC(=O)Nc2cc(C(=O)Nc3ccccc3)ccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.55
RARG P13631 5/20 0.55
RARA P10276 5/20 0.50
CYP26A1 O43174 4/20 0.50
CYP3A4 P08684 3/20 0.50
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
PTPN1 P18031 2/20 0.47
RORA P35398 1/20 0.46
RORC P51449 1/20 0.46
PLAU P00749 1/20 0.46
CYP26B1 Q9NR63 1/20 0.46
MAPT P10636 1/20 0.44
HDAC3 O15379 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9379480 0.88 BACE1 (0.52) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9376603 0.88 BACE1 (0.52) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9379462 0.86 RAB9A (0.53) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9376618 0.85 RARB (0.56) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9375662 0.84 MAPT (0.56) KMT2AMEN1MAPTRAB9APOLB
SCHEMBL23143565 0.82 TRPV1 (0.56) PTPN1RORARORCPLAUHDAC3
SCHEMBL9314264 0.81 MEN1 (0.53) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9312256 0.81 RARB (0.51) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9139650 0.81 RARB (0.73) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9312277 0.81 KMT2A (0.49) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0344634-B1 Bicyclic carboxamides, process for their preparation and medicaments containing them BOEHRINGER MANNHEIM GMBH (DE) 1994-03-30 EP disclosed
US-5019587-A Anticoagulants BOEHRINGER MANNHEIM GMBH (DE) 1991-05-28 US disclosed
WO-1991001986-A1 N-(DIALKYLOXOPHOSPHINYLALKYL)-LACTAMS, PROCESS FOR PREPARING THEM AND DRUGS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1991-02-21 WO disclosed