SCHEMBL9375261

SCHEMBL9375261

CC1(C)C(=O)Nc2cc(C(=O)Nc3ccc(F)cc3)ccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.55
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
CYP26A1 O43174 1/20 0.51
CYP3A4 P08684 1/20 0.51
RARA P10276 1/20 0.51
MAPT P10636 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TP53 P04637 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
POLB P06746 1/20 0.49
HTT P42858 1/20 0.49
PTPN1 P18031 1/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
ATM Q13315 1/20 0.48
MITF O75030 1/20 0.48
MAPK14 Q16539 3/20 0.47
SNCA P37840 1/20 0.47
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9380846 0.90 BACE1 (0.52) BACE1MEN1KMT2ACYP26A1CYP3A4
SCHEMBL9376571 0.88 CYP26A1 (0.52) BACE1MEN1KMT2ACYP26A1CYP3A4
SCHEMBL9375391 0.88 CYP26A1 (0.52) MEN1KMT2ACYP26A1CYP3A4RARA
SCHEMBL9380901 0.87 MEN1 (0.53) BACE1MEN1KMT2ACYP26A1CYP3A4
SCHEMBL9840186 0.87 CYP26A1 (0.51) BACE1MEN1KMT2ACYP26A1CYP3A4
SCHEMBL9379538 0.87 MEN1 (0.53) MEN1KMT2ACYP26A1CYP3A4RARA
SCHEMBL9374793 0.87 CYP26A1 (0.53) BACE1MEN1KMT2ACYP26A1CYP3A4
SCHEMBL9374775 0.86 NPC1 (0.52) MEN1KMT2AMAPTSMN1; SMN2NPC1
SCHEMBL9375240 0.86 KMT2A (0.52) MEN1KMT2ACYP26A1CYP3A4RARA
SCHEMBL9375945 0.85 MEN1 (0.54) MEN1KMT2ACYP26A1CYP3A4RARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0344634-B1 Bicyclic carboxamides, process for their preparation and medicaments containing them BOEHRINGER MANNHEIM GMBH (DE) 1994-03-30 EP claimed
WO-1991001986-A1 N-(DIALKYLOXOPHOSPHINYLALKYL)-LACTAMS, PROCESS FOR PREPARING THEM AND DRUGS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1991-02-21 WO disclosed