SCHEMBL9375288

SCHEMBL9375288

Clc1ccc(C2=CCN(CCCc3ccccc3)CC2)cc1

nearest known ligand 0.92

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 11/20 0.92
PARP1 P09874 2/20 0.60
HTR1A P08908 1/20 0.58
S1PR1 P21453 1/20 0.57
S1PR3 Q99500 1/20 0.57
DRD2 P14416 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9377531 0.96 SIGMAR1 (1.00) SIGMAR1PARP1HTR1AS1PR1S1PR3
Maleic Acid SCHEMBL8092718 0.87 SIGMAR1 (0.83) SIGMAR1PARP1HTR1AS1PR1S1PR3
Fumaric Acid SCHEMBL8092721 0.87 SIGMAR1 (0.83) SIGMAR1PARP1HTR1AS1PR1S1PR3
SCHEMBL10287534 0.84 SIGMAR1 (0.71) SIGMAR1HTR1ADRD2
SCHEMBL9473840 0.81 SIGMAR1 (0.92) SIGMAR1PARP1DRD2
SCHEMBL30484775 0.81 SIGMAR1 (0.66) SIGMAR1PARP1HTR1AS1PR1S1PR3
SCHEMBL11938943 0.80 SIGMAR1 (0.65) SIGMAR1HTR1ADRD2
SCHEMBL6626009 0.80 SIGMAR1 (0.65) SIGMAR1PARP1HTR1ADRD2
SCHEMBL5846298 0.80 SIGMAR1 (0.68) SIGMAR1PARP1HTR1ADRD2
SCHEMBL7289482 0.79 SIGMAR1 (0.67) SIGMAR1PARP1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP claimed
EP-0507863-A4 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF 1993-07-07 EP claimed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO claimed
EP-0507863-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1992-10-14 EP claimed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO claimed