SCHEMBL9375455

SCHEMBL9375455

COc1ccc(OC2=NC(C)(C)Oc3ccc(C#N)cc32)nn1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
ABCC9 O60706 3/20 0.31
BACE1 P56817 2/20 0.31
SCN9A Q15858 1/20 0.31
MALT1 Q9UDY8 1/20 0.31
OXTR P30559 1/20 0.31
AR P10275 1/20 0.30
TDP2 O95551 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9371377 0.90 ABCC9 (0.32) ABCC9
SCHEMBL9371892 0.85 ABCC9 (0.32) ABCC9
SCHEMBL9372051 0.82 DEGS1 (0.34) PDE4BABCC9SCN9AOXTR
SCHEMBL9371581 0.82 ABCC9 (0.36) ABCC9BACE1
SCHEMBL9373060 0.82 KDM4E (0.36) PDE4BABCC9BACE1SCN9A
SCHEMBL9372383 0.82 KDM4E (0.38) ABCC9OXTR
SCHEMBL9372537 0.81 ABCC9 (0.34) ABCC9
SCHEMBL9779754 0.81 ABCC9 (0.38) ABCC9
SCHEMBL9779615 0.81 ABCC9 (0.36) ABCC9SCN9A
SCHEMBL10435559 0.80 SMN1; SMN2 (0.35) ABCC9BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0371312-B1 Benzoxazine derivatives MERCK PATENT GMBH (DE) 1994-07-20 EP disclosed
US-5036068-A Cardiovascular disorders MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-07-30 US disclosed
EP-0371312-A1 Benzoxazine derivatives MERCK PATENT GmbH (DE) 1990-06-06 EP disclosed