SCHEMBL9779754

SCHEMBL9779754

CC1(C)N=C(Oc2cnccn2)c2cc(C#N)ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 3/20 0.38
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
PTGS2 P35354 2/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 2/20 0.32
POLB P06746 1/20 0.32
FNTA P49354 1/20 0.31
FNTB P49356 1/20 0.31
LTA4H P09960 1/20 0.31
TSHR P16473 1/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
FEN1 P39748 1/20 0.30
CYP19A1 P11511 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9372537 0.85 ABCC9 (0.34) ABCC9PTGS2
SCHEMBL9779615 0.84 ABCC9 (0.36) ABCC9
SCHEMBL9779813 0.81 ALK (0.38) ABCC9CYP11B1CYP11B2
SCHEMBL9371581 0.81 ABCC9 (0.36) ABCC9PTGS2
SCHEMBL9372051 0.81 DEGS1 (0.34) ABCC9FNTAFNTB
SCHEMBL9373060 0.81 KDM4E (0.36) ABCC9KDM4EPOLBALDH1A1FEN1
SCHEMBL9375455 0.81 PDE4A (0.33) ABCC9
SCHEMBL9371892 0.80 ABCC9 (0.32) ABCC9
SCHEMBL9779686 0.79 ABCC9 (0.32) ABCC9
SCHEMBL9372418 0.78 LMNA (0.39) ABCC9PTGS2MAPTKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5036068-A Cardiovascular disorders MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-07-30 US disclosed
EP-0371312-A1 Benzoxazine derivatives MERCK PATENT GmbH (DE) 1990-06-06 EP disclosed