SCHEMBL9375664

SCHEMBL9375664

CCc1ccn2c(C)c(CCc3ccc(N)c(O)c3)nc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
MEN1 O00255 2/20 0.37
GAA P10253 2/20 0.37
MAPT P10636 2/20 0.37
RAB9A P51151 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37
TRPA1 O75762 1/20 0.35
PRMT5 O14744 1/20 0.34
AKT1 P31749 1/20 0.32
AKT2 P31751 1/20 0.32
THRB P10828 1/20 0.32
ALDH1A1 P00352 2/20 0.31
GFER P55789 1/20 0.31
HTR6 P50406 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
SKP2 Q13309 1/20 0.31
USP7 Q93009 1/20 0.30
BACE1 P56817 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9376273 0.91 KDM4E (0.37) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9374989 0.88 KDM4E (0.39) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9377374 0.88 USP7 (0.41) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9380048 0.84 CREBBP (0.36) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9375832 0.84 KDM4E (0.39) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9376169 0.83 ALDH1A1 (0.42) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9376989 0.83 KMT2A (0.35) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9376914 0.83 PLAU (0.38) KDM4EGAAMAPTRAB9AAKT1
SCHEMBL9378823 0.79 NR1H4 (0.43) KDM4EMEN1GAAMAPTRAB9A
SCHEMBL9767536 0.79 KDM4E (0.39) KDM4EMEN1GAAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0356234-B1 New Benzazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1994-05-11 EP disclosed
US-5047411-A Antiulcer Agents, H2-Receptor Antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-09-10 US disclosed
EP-0356234-A2 New Benzazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed