SCHEMBL9375670

SCHEMBL9375670

COc1ccn2c(C)c(CCc3ccc4nc(N)sc4c3)nc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C19 P33261 1/20 0.51
RAB9A P51151 3/20 0.45
NPC1 O15118 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 2/20 0.42
KCNH2 Q12809 3/20 0.41
DRD2 P14416 2/20 0.41
TSHR P16473 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
APP P05067 2/20 0.38
PIK3CA P42336 3/20 0.38
PI4KA P42356 3/20 0.38
PIK3CG P48736 3/20 0.38
PI4KB Q9UBF8 3/20 0.38
PIK3CD O00329 2/20 0.38
PIK3CB P42338 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9375280 0.87 RAB9A (0.49) CYP3A4CYP1A2CYP2C19RAB9ANPC1
Hydrochloric Acid SCHEMBL9383081 0.84 RAB9A (0.46) CYP3A4CYP1A2CYP2C19RAB9ANPC1
SCHEMBL9379336 0.82 NPC1 (0.57) CYP3A4CYP1A2CYP2C19RAB9ANPC1
SCHEMBL9378131 0.82 CREBBP (0.38) RAB9AALDH1A1
SCHEMBL9376391 0.81 CYP19A1 (0.48) RAB9ANPC1ALDH1A1TP53
SCHEMBL9379863 0.80 CREBBP (0.36) RAB9ANPC1SMN1; SMN2MAPTPIK3CG
SCHEMBL9375832 0.79 KDM4E (0.39) CYP3A4CYP1A2RAB9AMAPTTSHR
Hydrochloric Acid SCHEMBL9377697 0.79 CREBBP (0.36) RAB9AMAPTALDH1A1PIK3CG
SCHEMBL9376418 0.78 RAB9A (0.48) CYP3A4CYP1A2CYP2C19RAB9ANPC1
SCHEMBL9376180 0.78 TYMS (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0356234-B1 New Benzazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1994-05-11 EP disclosed
US-5047411-A Antiulcer Agents, H2-Receptor Antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-09-10 US disclosed
EP-0356234-A2 New Benzazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed