SCHEMBL9375677

SCHEMBL9375677

O=C(Nc1cccnc1N1CCNCC1)C(F)(F)F.O=C(OCc1ccccc1)N1CCN(c2ncccc2NC(=O)C(F)(F)F)CC1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 1/20 0.51
GRIN2B Q13224 12/20 0.48
HDAC1 Q13547 1/20 0.47
CYP2D6 P10635 4/20 0.41
CYP2C9 P11712 4/20 0.41
CYP3A4 P08684 3/20 0.41
TGM2 P21980 1/20 0.40
EPHX2 P34913 1/20 0.40
TRPA1 O75762 1/20 0.40
HSD11B1 P28845 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8924252 0.94 HDAC1 (0.52) SLC29A1GRIN2BHDAC1CYP2D6CYP2C9
SCHEMBL8918450 0.83 EPHX2 (0.56) EPHX2
SCHEMBL8923780 0.82 HDAC1 (0.52) SLC29A1GRIN2BHDAC1CYP2D6CYP2C9
SCHEMBL9376237 0.79 EPHX2 (0.48) EPHX2
SCHEMBL2088315 0.76 ACHE (0.52) HDAC1TGM2
SCHEMBL8917544 0.76 HDAC1 (0.49) SLC29A1GRIN2BHDAC1CYP2D6CYP2C9
Trifluoroacetic Acid SCHEMBL31505451 0.75 MEN1 (0.54) SLC29A1GRIN2BCYP2D6CYP2C9TGM2
Trifluoroacetic Acid SCHEMBL31505483 0.75 MEN1 (0.57) SLC29A1GRIN2BCYP2D6CYP2C9
Trifluoroacetic Acid SCHEMBL27706408 0.75 MEN1 (0.57) SLC29A1GRIN2BCYP2D6CYP2C9
SCHEMBL8921825 0.74 HDAC1 (0.58) SLC29A1GRIN2BHDAC1CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0594702-A1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS. UPJOHN CO (US) 1994-05-04 EP disclosed
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed