SCHEMBL9376162

SCHEMBL9376162

O=C1c2ccccc2CN1CCCCN1CCC(c2nsc3ccccc23)CC1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.58
HTR1A P08908 2/20 0.58
HTR2A P28223 1/20 0.58
DRD5 P21918 2/20 0.52
DRD3 P35462 2/20 0.52
HTR7 P34969 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9380479 0.99 DRD2 (0.58) DRD2HTR1AHTR2ADRD5DRD3
SCHEMBL9377355 0.84 HTR1A (0.65) DRD2HTR1AHTR2ADRD3HTR7
Hydrochloric Acid SCHEMBL9381340 0.82 HTR1A (0.62) DRD2HTR1AHTR2ADRD3HTR7
SCHEMBL9601759 0.82 HTR1A (0.70) DRD2HTR1AHTR2AHTR7
SCHEMBL30649298 0.82 HTR1A (0.70) DRD2HTR1AHTR2AHTR7
Hydrochloric Acid SCHEMBL9382359 0.81 HTR1A (0.69) DRD2HTR1AHTR2AHTR7
Hydrochloric Acid SCHEMBL9595406 0.80 HTR1A (0.71) DRD2HTR1AHTR2AHTR7
Hydrochloric Acid SCHEMBL9379578 0.80 HTR1A (0.71) DRD2HTR1AHTR2AHTR7
Hydrochloric Acid SCHEMBL9376327 0.79 HTR1A (0.66) DRD2HTR1AHTR2AHTR7
SCHEMBL9377459 0.78 DRD2 (0.55) DRD2HTR1AHTR2ADRD3HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625978-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS THE WELLCOME FOUNDATION LIMITED (GB) 1994-11-30 EP disclosed