SCHEMBL9376753

SCHEMBL9376753

CC1(C)N=C(n2cccc(Cl)c2=O)c2cc(C#N)ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 12/20 0.38
NPBWR1 P48145 1/20 0.33
MCHR1 Q99705 1/20 0.33
MALT1 Q9UDY8 1/20 0.33
ABCB1 P08183 2/20 0.32
BACE1 P56817 2/20 0.32
ICMT O60725 1/20 0.32
CTSD P07339 1/20 0.32
CASP3 P42574 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779700 0.87 ABCC9 (0.37) ABCC9MALT1ABCB1BACE1CTSD
SCHEMBL9374699 0.87 ABCC9 (0.37) ABCC9MALT1ABCB1BACE1CTSD
SCHEMBL9372600 0.86 ABCC9 (0.39) ABCC9MALT1ABCB1
SCHEMBL9377387 0.85 PDE4A (0.38) ABCC9NPBWR1MCHR1BACE1ICMT
SCHEMBL9373199 0.84 ABCC9 (0.36) ABCC9MALT1ABCB1BACE1CTSD
SCHEMBL9378100 0.84 ABCC9 (0.36) ABCC9MALT1ABCB1
SCHEMBL9372849 0.84 ABCC9 (0.36) ABCC9MALT1ABCB1BACE1CTSD
SCHEMBL9372282 0.83 ABCC9 (0.38) ABCC9MALT1ABCB1BACE1
SCHEMBL9779684 0.83 ABCC9 (0.37) ABCC9MALT1ABCB1BACE1ICMT
SCHEMBL9379748 0.83 ABCC9 (0.35) ABCC9MALT1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0371312-B1 Benzoxazine derivatives MERCK PATENT GMBH (DE) 1994-07-20 EP disclosed
US-5036068-A Cardiovascular disorders MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-07-30 US disclosed
EP-0371312-A1 Benzoxazine derivatives MERCK PATENT GmbH (DE) 1990-06-06 EP disclosed