SCHEMBL9379643

SCHEMBL9379643

CCNc1ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TYMS P04818 4/20 0.56
GART P22102 2/20 0.55
CA2 P00918 3/20 0.47
CA1 P00915 2/20 0.47
NAALAD2 Q9Y3Q0 2/20 0.45
FOLR1 P15328 6/20 0.45
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
FOLR2 P14207 3/20 0.43
ATIC P31939 2/20 0.43
SLC19A1 P41440 2/20 0.43
SLC46A1 Q96NT5 2/20 0.43
DHFR P00374 1/20 0.43
EHMT2 Q96KQ7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9379640 1.00 TYMS (0.56) TYMSGARTCA2CA1NAALAD2
SCHEMBL27513231 0.90 TYMS (0.55) TYMSGARTCA2CA1NAALAD2
SCHEMBL9829787 0.90 TYMS (0.55) TYMSGARTCA2CA1NAALAD2
SCHEMBL9829799 0.90 TYMS (0.55) TYMSGARTCA2CA1NAALAD2
SCHEMBL9828671 0.86 TYMS (0.53) TYMSGARTCA2CA1NAALAD2
SCHEMBL9828665 0.86 TYMS (0.53) TYMSGARTCA2CA1NAALAD2
SCHEMBL27559568 0.81 CA2 (0.53) GARTCA2CA1NAALAD2FOLR1
SCHEMBL9600674 0.80 CA2 (0.52) TYMSGARTCA2CA1NAALAD2
SCHEMBL9600688 0.80 CA2 (0.52) TYMSGARTCA2CA1NAALAD2
SCHEMBL9555966 0.78 L3MBTL1 (0.51) TYMSGARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0318225-B1 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents ICI PLC (GB) 1994-03-16 EP disclosed
EP-0239362-B1 ANTI-TUMOR AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-12-04 EP disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed
EP-0239362-A2 Anti-tumor agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-09-30 EP disclosed