SCHEMBL9380372

SCHEMBL9380372

NCCCCN1CCN(c2csc3ccccc23)CC1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.50
DRD2 P14416 5/20 0.50
HTR2A P28223 3/20 0.50
CYP2D6 P10635 1/20 0.49
SIGMAR1 Q99720 1/20 0.48
DRD3 P35462 2/20 0.47
SLC6A4 P31645 1/20 0.46
ADRA1A P35348 1/20 0.46
HRH1 P35367 1/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573898 0.83 DRD2 (0.67) HTR1ADRD2HTR2AADRA1AHRH1
SCHEMBL7815509 0.82 HTR2A (0.61) HTR1ADRD2HTR2AADRA1A
SCHEMBL9381448 0.81 HTR1A (0.76) HTR1ADRD2HTR2ACYP2D6DRD3
Hydrochloric Acid SCHEMBL9380816 0.80 HTR1A (0.74) HTR1ADRD2HTR2ADRD3
SCHEMBL4307891 0.79 DRD4 (0.46) DRD2HTR2ASIGMAR1DRD3ADRA1A
SCHEMBL4299920 0.78 HTR2A (0.57) HTR1ADRD2HTR2AADRA1A
Hydrochloric Acid SCHEMBL4307355 0.78 DRD4 (0.46) HTR2ASIGMAR1ADRA1A
SCHEMBL4310830 0.78 DRD4 (0.46) DRD2HTR2ASIGMAR1DRD3ADRA1A
SCHEMBL4438394 0.78 HTR2A (0.56) HTR1ADRD2HTR2AADRA1A
SCHEMBL3122433 0.76 SLC6A4 (0.70) HTR1ADRD2SIGMAR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625978-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS THE WELLCOME FOUNDATION LIMITED (GB) 1994-11-30 EP disclosed
WO-1993016073-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS THE WELLCOME FOUNDATION LIMITED (GB) 1993-08-19 WO disclosed