SCHEMBL9380765

SCHEMBL9380765

CN(C)C(=S)c1ccc2cc(Br)ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 3/20 0.47
ALDH1A1 P00352 6/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
BACE1 P56817 1/20 0.47
MAPT P10636 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2A6 P11509 1/20 0.42
KDM4E B2RXH2 1/20 0.39
LMNA P02545 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
DHODH Q02127 2/20 0.37
F10 P00742 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29636491 0.81 ALDH1A1 (0.57) ALDH1A1HPGDHSD17B10CYP2C9CYP2C19
SCHEMBL6703588 0.80 ALDH1A1 (0.60) ALDH1A1HPGDHSD17B10CYP2C9CYP2C19
SCHEMBL11053906 0.79 NCEH1 (0.43) NCEH1ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL11049872 0.76 NCEH1 (0.43) NCEH1ALDH1A1HPGDMEN1KMT2A
SCHEMBL15644255 0.75 ALDH1A1 (0.48) NCEH1ALDH1A1BACE1MAPTMEN1
SCHEMBL4072743 0.71 NCEH1 (0.66) NCEH1ALDH1A1CYP2C9CYP2C19MAPT
SCHEMBL264367 0.71 CYP2A6 (0.55) NCEH1ALDH1A1HPGDMAPTMEN1
SCHEMBL30350490 0.71 CYP2A6 (0.55) NCEH1ALDH1A1HPGDMAPTMEN1
SCHEMBL2643193 0.71 CYP2A6 (0.46) NCEH1ALDH1A1BACE1MAPTMEN1
SCHEMBL29353067 0.69 CYP2A6 (0.77) NCEH1ALDH1A1CYP2C19BACE1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0409413-B1 Diaryl ether heterocycles ICI PLC (GB) 1994-08-03 EP disclosed
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed
EP-0409413-A2 Diaryl ether heterocycles IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed