SCHEMBL9385274

SCHEMBL9385274

COc1ccn2c3c(cc2c1)CC(CO)CC3

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 1/20 0.39
MAPT P10636 1/20 0.37
CYP19A1 P11511 3/20 0.37
SIGMAR1 Q99720 2/20 0.35
HTR1A P08908 1/20 0.35
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
BAZ2B Q9UIF8 1/20 0.33
BAZ2A Q9UIF9 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
MCHR1 Q99705 1/20 0.32
OPRK1 P41145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9386696 0.84 MTNR1A (0.36) CYP26A1MAPTCYP19A1SIGMAR1HTR1A
SCHEMBL1991216 0.79 GBA1 (0.33) MAPTCYP19A1SIGMAR1HTR1A
SCHEMBL8318762 0.79 GBA1 (0.33) MAPTCYP19A1SIGMAR1HTR1A
SCHEMBL8324468 0.79 GBA1 (0.33) MAPTCYP19A1SIGMAR1HTR1A
SCHEMBL4623036 0.73 CYP26A1 (0.67) CYP26A1CYP19A1SIGMAR1HTR1ADRD2
SCHEMBL9630417 0.73 CYP19A1 (0.63) CYP26A1CYP19A1SIGMAR1HTR1ADRD2
SCHEMBL7288575 0.73 CYP26A1 (0.67) CYP26A1CYP19A1SIGMAR1HTR1ADRD2
Trifluoromethanesulfonic Acid SCHEMBL9419763 0.67 CYP26A1 (0.55) CYP26A1CYP19A1SIGMAR1DRD2DRD3
SCHEMBL6015851 0.66 HTT (0.38) MAPTMCHR1OPRK1
SCHEMBL8319230 0.66 HTT (0.38) MAPTMCHR1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0384349-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1994-04-27 EP disclosed