SCHEMBL8318762

SCHEMBL8318762

OC[C@H]1CCc2c(cc3ccccn23)C1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
HTR1A P08908 2/20 0.31
SIGMAR1 Q99720 2/20 0.31
CYP19A1 P11511 1/20 0.31
THRB P10828 1/20 0.30
CYP2D6 P10635 1/20 0.30
HTT P42858 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1991216 1.00 GBA1 (0.33) GBA1L3MBTL1NPC1MAPTRAB9A
SCHEMBL8324468 1.00 GBA1 (0.33) GBA1L3MBTL1NPC1MAPTRAB9A
SCHEMBL9387801 0.85 SLC6A2 (0.32) HTR1ASIGMAR1CYP19A1
SCHEMBL8449850 0.83 DGAT1 (0.45) MAPT
SCHEMBL8319230 0.79 HTT (0.38) L3MBTL1NPC1MAPTRAB9AHTT
SCHEMBL6015851 0.79 HTT (0.38) L3MBTL1NPC1MAPTRAB9AHTT
SCHEMBL9385274 0.79 CYP26A1 (0.39) MAPTHTR1ASIGMAR1CYP19A1
SCHEMBL9385160 0.77 L3MBTL1 (0.34) GBA1L3MBTL1NPC1MAPTRAB9A
SCHEMBL1999145 0.77 BUB1 (0.32) L3MBTL1HTTATM
SCHEMBL8452787 0.75 TBXAS1 (0.36) L3MBTL1NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574783-B1 Asymmetric hydrogenation HOFFMANN LA ROCHE (CH) 1999-10-06 EP claimed
US-5374727-A Using rhodium-diphosphine complex as hydrogenation catalyst HOFFMANN-LA ROCHE INC. (US) 1994-12-20 US claimed
EP-0574783-A2 Asymmetric hydrogenation F. HOFFMANN-LA ROCHE AG (CH) 1993-12-22 EP claimed
EP-0574783-B1 Asymmetric hydrogenation HOFFMANN LA ROCHE (CH) 1999-10-06 EP disclosed
EP-0624586-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-09-01 EP disclosed
EP-0540956-B1 Process for the manufacture of substituted maleimides HOFFMANN LA ROCHE (CH) 1997-09-03 EP disclosed
US-5399712-A Protein kinase C inhibitor HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
US-5374727-A Using rhodium-diphosphine complex as hydrogenation catalyst HOFFMANN-LA ROCHE INC. (US) 1994-12-20 US disclosed
EP-0624586-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1994-11-17 EP disclosed
EP-0574783-A2 Asymmetric hydrogenation F. HOFFMANN-LA ROCHE AG (CH) 1993-12-22 EP disclosed
EP-0540956-A1 Process for the manufacture of substituted maleimides F. HOFFMANN-LA ROCHE AG (CH) 1993-05-12 EP disclosed