SCHEMBL9388336

SCHEMBL9388336

O=C(C1=CC=Cc2ccccc2N1)c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 2/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
LMNA P02545 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
NAPRT Q6XQN6 1/20 0.40
P4HTM Q9NXG6 1/20 0.40
ALDH1A1 P00352 3/20 0.39
TSHR P16473 1/20 0.38
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
GSK3B P49841 1/20 0.36
HSD17B14 Q9BPX1 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
TGM2 P21980 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29013777 0.78 MAPT (0.42) KMT2AKDM4ELMNAL3MBTL1NAPRT
SCHEMBL28619553 0.77 ALDH1A1 (0.38) KMT2AKDM4ELMNAALDH1A1MAPT
SCHEMBL8330072 0.76 MAPT (0.47) KMT2AKDM4ELMNANAPRTALDH1A1
SCHEMBL14691822 0.74 MAPT (0.45) KMT2ALMNAALDH1A1MAPTGAA
Hydrochloric Acid SCHEMBL8332139 0.74 MAPT (0.45) KMT2AKDM4ELMNANAPRTALDH1A1
SCHEMBL858689 0.74 MAPT (0.45) LMNAL3MBTL1TSHRMAPTGAA
SCHEMBL8672572 0.73 MAPT (0.38) KMT2ALMNAALDH1A1MAPTGAA
SCHEMBL9935617 0.71 MAPT (0.54) MAPTGAARAB9A
SCHEMBL28529505 0.71 MAPT (0.41) KMT2AKDM4EALDH1A1MAPTGAA
SCHEMBL28880924 0.69 MAPT (0.42) KDM4ELMNAL3MBTL1P4HTMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994014796-A1 NOVEL N-(PYRIDYLCARBONYL)BENZAZEPINE DERIVATIVE AND INTERMEDIATE THEREFOR YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-07-07 WO disclosed