SCHEMBL9388387

SCHEMBL9388387

Cn1c(N2CCN(CCCOc3ccc([N+](=O)[O-])cc3O)CC2)cc(=O)n(C)c1=O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.46
HTR2A P28223 3/20 0.46
HRH1 P35367 2/20 0.43
HRH2 P25021 1/20 0.43
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
PKM P14618 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
MAPT P10636 2/20 0.40
GALR3 O60755 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9385389 0.99 HTR1A (0.46) HTR1AHTR2AHRH1HRH2ALDH1A1
SCHEMBL9385200 0.92 HTR1A (0.45) HTR1AHTR2AHRH1HRH2ALDH1A1
Hydrochloric Acid SCHEMBL9384750 0.91 HTR1A (0.44) HTR1AHTR2AHRH1HRH2ALDH1A1
SCHEMBL9388176 0.88 HTR1A (0.45) HTR1AHTR2AHRH1ALDH1A1SMN1; SMN2
SCHEMBL9383653 0.88 MAPT (0.48) HTR1AHTR2AALDH1A1SMN1; SMN2PKM
SCHEMBL9384567 0.88 HTR1A (0.45) HTR1AHTR2AHRH1HRH2ALDH1A1
SCHEMBL9386908 0.88 HTR1A (0.45) HTR1AHTR2AHRH1ALDH1A1SMN1; SMN2
SCHEMBL9384577 0.88 HTR1A (0.46) HTR1AHTR2AHRH1HRH2ALDH1A1
SCHEMBL9388964 0.88 HTR1A (0.50) HTR1AHTR2AHRH1HRH2ALDH1A1
Hydrochloric Acid SCHEMBL9385657 0.87 MAPT (0.44) HTR1AHTR2AHRH1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0369627-B1 Pyrimidinedione derivative compounds, method of producing the same and antiarrythmic agents containing the same MITSUI TOATSU CHEMICALS (JP) 1994-12-21 EP disclosed
US-5008267-A Pyrimidinedione compounds, method of producing the same and antiarrythmic agents containing the same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1991-04-16 US disclosed
EP-0369627-A2 Pyrimidinedione derivative compounds, method of producing the same and antiarrythmic agents containing the same MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-05-23 EP disclosed