SCHEMBL9389409

SCHEMBL9389409

CCc1ccc2c(=O)cc(O)c(=O)[nH]c2c1

nearest known ligand 0.78

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DAO P14920 7/20 0.68
DDO Q99489 3/20 0.51
KIF11 P52732 1/20 0.49
CDK1 P06493 1/20 0.46
CDK2 P24941 1/20 0.46
CTSV O60911 1/20 0.44
CTSL P07711 1/20 0.44
PTGES O14684 1/20 0.43
CYP2C9 P11712 1/20 0.43
TRPA1 O75762 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9389933 0.88 DAO (0.52) DAODDOCTSVCTSLPTGES
SCHEMBL9393070 0.88 DAO (0.63) DAODDOKIF11CTSVCTSL
SCHEMBL16767852 0.81 DAO (1.00) DAODDOTRPA1
SCHEMBL19032120 0.79 LMNA (0.60) DAOKIF11CTSVCTSL
SCHEMBL9387604 0.79 DAO (0.55) DAODDO
SCHEMBL9387738 0.79 DAO (0.65) DAODDOKIF11
SCHEMBL13267221 0.78 KDM4E (0.54) DAOKIF11CDK1CDK2TRPA1
SCHEMBL9452268 0.77 KDM4E (0.61) KIF11CYP2C9
SCHEMBL9389308 0.76 DAO (0.56) DAODDO
SCHEMBL9393210 0.76 DAO (0.49) DAODDO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed