SCHEMBL9389842

SCHEMBL9389842

Cc1cc2c(=O)cc(O)c(=O)[nH]c2cc1Br

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.47
DDO Q99489 2/20 0.47
GSK3B P49841 4/20 0.45
CCNB2 O95067 2/20 0.41
CDK1 P06493 2/20 0.41
CCNB1 P14635 2/20 0.41
GSK3A P49840 2/20 0.41
CDK5 Q00535 2/20 0.41
CDK5R1 Q15078 2/20 0.41
CCNB3 Q8WWL7 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
SRC P12931 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352458 0.86 DAO (0.53) DAODDOKDM4EALDH1A1GLA
SCHEMBL9389319 0.81 GRIN2D (0.56) DAODDOKDM4EALDH1A1MAPT
SCHEMBL9388916 0.74 KDM4E (0.46) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL9393064 0.74 DAO (0.36) DAODDOSRC
SCHEMBL9007836 0.73 METAP2 (0.49) DAODDOGSK3BCCNB2CDK1
SCHEMBL9387730 0.73 HPGD (0.60) DAODDOGSK3BCDK1CCNB1
SCHEMBL9387604 0.73 DAO (0.55) DAODDOSRC
SCHEMBL9387738 0.73 DAO (0.65) DAODDOKDM4EALDH1A1
SCHEMBL9387632 0.73 DAO (0.65) DAODDOKDM4EALDH1A1MAPT
SCHEMBL9387925 0.73 DAO (0.53) DAODDOSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed