Penfluridol

Penfluridol

SCHEMBL93939

OC1(c2ccc(Cl)c(C(F)(F)F)c2)CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 11/20 1.00
DRD2 P14416 10/20 1.00
OPRK1 P41145 8/20 1.00
DRD3 P35462 8/20 1.00
HTR1A P08908 7/20 1.00
DRD4 P21917 7/20 1.00
HTR2A P28223 7/20 1.00
HTR2C P28335 7/20 1.00
HTR7 P34969 7/20 1.00
HTR1D P28221 6/20 1.00
HRH2 P25021 6/20 1.00
HTR2B P41595 6/20 1.00
OPRD1 P41143 6/20 1.00
DRD1 P21728 5/20 1.00
DRD5 P21918 5/20 1.00
SLC6A2 P23975 5/20 1.00
SLC6A4 P31645 5/20 1.00
HTR6 P50406 5/20 1.00
SLC6A3 Q01959 5/20 1.00
HRH1 P35367 4/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Penfluridol SCHEMBL30546621 1.00 OPRM1 (1.00) OPRM1DRD2OPRK1DRD3HTR1A
Penfluridol SCHEMBL28123335 0.97 OPRM1 (0.94) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL905023 0.97 OPRM1 (1.00) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL904950 0.94 OPRM1 (0.89) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL905043 0.93 OPRM1 (0.87) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL905046 0.92 OPRM1 (0.85) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL905028 0.92 OPRM1 (1.00) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL904992 0.91 OPRM1 (0.84) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL905031 0.89 OPRM1 (0.81) OPRM1DRD2OPRK1DRD3HTR1A
SCHEMBL905064 0.89 OPRM1 (0.84) OPRM1DRD2OPRK1DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3424 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12550885-B2 Red blood cell storage solutions, solution additives, and methods for improving the storage of red blood cells UNIVERSITY OF CINCINNATI (US) 2026-02-17 US claimed
EP-3507371-B1 COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM UNIV RUTGERS (US) 2026-01-28 EP claimed
US-12527754-B2 Methods and compositions for preventing and treating metabolic syndrome induced by antipsychotic treatment and related diseases and conditions TUFTS MEDICAL CENTER, INC. (US) 2026-01-20 US claimed
EP-4658278-A1 SELECTIVE FIASMA TREATMENT Valo Health, Inc. (US) 2025-12-10 EP claimed
EP-3625238-B1 NOVEL SPIRO-LACTAM COMPOUNDS, PROCESS AND USES THEREOF UNIV DE COIMBRA (PT) 2025-11-26 EP claimed
EP-4618973-A1 METHODS OF SWITCHING NEUROPSYCHIATRIC MEDICATIONS USING ULOTARONT Sumitomo Pharma America, Inc. (US) 2025-09-24 EP claimed
US-20250262167-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2025-08-21 US claimed
US-20250179064-A1 BENZOQUINOLONE INHIBITORS OF VMAT2 AUSPEX PHARMACEUTICALS LLC 2025-06-05 US claimed
US-20250170143-A1 METHODS OF TREATING OCULAR FIBROTIC PATHOLOGIES MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2025-05-29 US claimed
WO-2025101418-A1 TREATMENT OF PSYCHIATRIC OR NEUROLOGICAL DISORDERS IN PATIENTS WITH PROMINENT ANHEDONIA USING IRDABISANT AS A MONOTHERAPY OR IN COMBINATION WITH AN ANTIPSYCHOTIC AGENT ALTO NEUROSCIENCE, INC. (US) 2025-05-15 WO claimed
WO-1998043646-A1 NEW THERAPEUTIC COMBINATIONS OF MIRTAZAPINE AND ANTIPSYCHOTIC AGENTS, FOR THE TREATMENT OR PROPHYLAXIS OF PSYCHOTIC DISORDERS AKZO NOBEL N.V. (NL) 1998-10-08 WO claimed
WO-1996001631-A1 NOVEL COMBINATION PRODUCT COMPRISING CAPRIPRAMINE AND A NEUROLEPTIC PIERRE FABRE MEDICAMENT (FR) 1996-01-25 WO claimed
WO-1994023726-A1 CALMODULIN BLOCKING AGENT ADDUCTS USEFUL AS ANTI-PLATELET AGENTS MALLINCKRODT MEDICAL, INC. (US) 1994-10-27 WO claimed
US-4654323-A BLOCKING AGENT FOR CALCIUM CALMODULIN COMPLEX BAR ILAN UNIVERSITY (IL) 1987-03-31 US claimed
US-4443446-A Use of psychoactive drugs as vaginal contraceptives UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1984-04-17 US claimed
EP-0082203-A1 USE OF CALMODULIN BINDING DRUGS IN UTERUS TO PREVENT PREGNANCY THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1983-06-29 EP claimed
US-4377577-A Use of psychoactive drugs in uterus to prevent pregnancy UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1983-03-22 US claimed
WO-1983000086-A1 USE OF CALMODULIN BINDING DRUGS IN UTERUS TO PREVENT PREGNANCY UNIV GEORGIA RES FOUND (US) 1983-01-20 WO claimed
EP-0053108-A1 VAGINAL CONTRACEPTIVES COMPRISING PSYCHOACTIVE DRUGS THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1982-06-09 EP claimed
WO-1981003421-A1 USE OF PSYCHOACTIVE DRUGS AS VAGINAL CONTRACEPTIVES UNIV GEORGIA (US) 1981-12-10 WO claimed