SCHEMBL9397459

SCHEMBL9397459

CCCCCN1CC[C@H](c2ccccc2)[C@@H](COc2ccc3c(c2)OCO3)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.54
L3MBTL1 Q9Y468 1/20 0.51
CYP3A4 P08684 5/20 0.47
CYP1A2 P05177 3/20 0.47
CYP2D6 P10635 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
CYP2C9 P11712 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
MAPK1 P28482 2/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
SLC6A4 P31645 2/20 0.46
TP53 P04637 2/20 0.46
GRK2 P25098 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NPC1 O15118 1/20 0.46
CACNA1F O60840 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9397596 1.00 HTR1A (0.54) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
SCHEMBL9397462 1.00 HTR1A (0.54) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL1152347 0.99 HTR1A (0.54) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL1152345 0.99 HTR1A (0.54) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
SCHEMBL10431404 0.97 HTR1A (0.53) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
SCHEMBL10431405 0.97 HTR1A (0.53) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
SCHEMBL8604020 0.92 L3MBTL1 (0.53) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
SCHEMBL8604024 0.92 L3MBTL1 (0.53) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
SCHEMBL1151876 0.91 L3MBTL1 (0.63) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6
SCHEMBL7413959 0.91 L3MBTL1 (0.52) HTR1AL3MBTL1CYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266574-B1 Piperidine compounds and their preparation and use NOVO NORDISK AS (DK) 1994-01-05 EP claimed
EP-0374675-A2 Reduction of piperidine-dion-derivatives and intermediates NOVO NORDISK A/S (DK) 1990-06-27 EP disclosed