SCHEMBL9399457

SCHEMBL9399457

CC(C)(Nc1ccnc2ccccc12)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.51
PTPN11 Q06124 1/20 0.51
HTR1A P08908 2/20 0.49
ADRA1D P25100 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
HTR2C P28335 3/20 0.47
HTR2B P41595 3/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC3 O15379 1/20 0.47
ACHE P22303 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
DNMT1 P26358 1/20 0.47
DNMT3L Q9UJW3 1/20 0.47
DNMT3A Q9Y6K1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9400132 0.85 PTPN1 (0.49) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL13230464 0.80 HTR1A (0.58) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL5176476 0.77 CYP1A2 (0.48) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL7370108 0.76 PTPN1 (0.67) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL1695394 0.75 CACNA2D1 (0.52) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL7504880 0.75 HTR1A (0.51) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL13113090 0.74 MEN1 (0.79) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL4474966 0.74 HTR1A (0.54) PTPN1PTPN11HTR1AADRA1DADRA1A
SCHEMBL329187 0.74 KDM4E (0.51) MEN1KMT2AGSK3BKDM4EALDH1A1
SCHEMBL27297227 0.74 HTR1A (0.58) PTPN1PTPN11HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5331006-A Cholecystokinin, antisecretory agents WARNER-LAMBERT COMPANY (US) 1994-07-19 US disclosed
WO-1992004025-A1 AMINO ACID ANALOGS AS CCK ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1992-03-19 WO disclosed