SCHEMBL9401778

SCHEMBL9401778

CC1=C(C(=O)O)C(c2cccc([N+](=O)[O-])c2)C(C(=O)O)=C(C)N1CCC=CC=Cc1ccc(Cn2ccnc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.43
CYP17A1 P05093 2/20 0.43
CYP21A2 P08686 2/20 0.43
CYP19A1 P11511 5/20 0.42
TBXAS1 P24557 5/20 0.42
CYP1A2 P05177 3/20 0.42
LMNA P02545 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
USP2 O75604 1/20 0.42
CACNA1B Q00975 2/20 0.41
TP53 P04637 1/20 0.39
MDM2 Q00987 1/20 0.39
CYP11B2 P19099 2/20 0.38
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401777 0.95 CYP11B1 (0.44) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401775 0.86 CACNA1B (0.51) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401787 0.86 CACNA1B (0.51) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401791 0.83 CYP17A1 (0.41) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401783 0.82 CACNA1B (0.56) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401773 0.82 CACNA1B (0.56) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401969 0.81 CACNA1B (0.56) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401782 0.81 CACNA1B (0.56) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9401841 0.81 CACNA1B (0.56) CYP11B1CYP17A1CYP21A2CYP19A1TBXAS1
SCHEMBL9833247 0.79 CACNA1B (0.59) CYP1A2LMNACYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286869-A Vasodilators and anticoagulants FUJIREBIO KABUSHIKI KAISHA (JP) 1994-02-15 US disclosed
EP-0403957-A2 Optical active 1,4-dihydropyridine derivates FUJIREBIO INC. (JP) 1990-12-27 EP disclosed