SCHEMBL9833247

SCHEMBL9833247

CC1=C(C(=O)O)C(c2cccc([N+](=O)[O-])c2)C(C(=O)O)=C(C)N1CCC=Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.59
CACNA1C Q13936 5/20 0.52
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.52
ADORA3 P0DMS8 2/20 0.52
HTT P42858 2/20 0.52
MLNR O43193 1/20 0.52
NR1I2 O75469 1/20 0.52
CACNA1H O95180 1/20 0.52
NR3C1 P04150 1/20 0.52
TBXA2R P21731 1/20 0.52
PDE4D Q08499 1/20 0.52
SLC29A1 Q99808 1/20 0.52
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 3/20 0.47
CYP2C19 P33261 3/20 0.47
MAPT P10636 3/20 0.47
CYP2D6 P10635 2/20 0.47
TSHR P16473 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401777 0.84 CYP11B1 (0.44) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL3443986 0.84 CYP1A2 (0.55) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL30873727 0.81 CYP1A2 (0.57) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL5396699 0.81 CYP1A2 (0.48) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL5396705 0.81 CYP1A2 (0.48) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL20801670 0.81 CYP1A2 (0.55) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL8403732 0.80 MAPT (0.50) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL28408223 0.80 LMNA (0.58) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL6534522 0.80 CACNA1C (0.69) CACNA1BCACNA1CKMT2AMEN1ADORA3
SCHEMBL10656803 0.80 CACNA1F (0.53) CACNA1BCACNA1CKMT2AMEN1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161877-B1 1,4-DIHYDROPYRIDINE DERIVATIVES, METHODS FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME FUJIREBIO KABUSHIKI KAISHA also trading as FUJIREBIO INC. (JP) 1991-05-29 EP claimed