SCHEMBL9404072

SCHEMBL9404072

Nc1cc(S(=O)(=O)CCO)ccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.55
MAPT P10636 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 1/20 0.43
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA9 Q16790 3/20 0.41
CA7 P43166 2/20 0.41
CA14 Q9ULX7 2/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
LOX P28300 1/20 0.40
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
CCR2 P41597 1/20 0.39
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9498638 0.86 CA2 (0.58) CA2POLBCA12CA1CA9
SCHEMBL8951864 0.84 MAPT (0.45) CA2MAPTNPSR1CA12CA1
SCHEMBL7029931 0.84 CA2 (0.53) CA2POLBLOXCCR2MEN1
SCHEMBL3369801 0.84 CA2 (0.60) CA2MAPTPOLBCA12CA1
SCHEMBL9178626 0.81 MAPT (0.40) CA2MAPTNPSR1CA12CA1
SCHEMBL5677264 0.81 CA2 (0.61) CA2MAPTPOLBCA12CA1
SCHEMBL10606415 0.81 CA2 (0.81) CA2MAPTPOLBCA12CA1
SCHEMBL10693250 0.80 GAA (0.52) CA2MAPTNPSR1POLBCA12
SCHEMBL11400330 0.80 MAPT (0.47) CA2MAPTNPSR1CA12CA1
SCHEMBL11323062 0.80 CA2 (0.43) CA2MAPTNPSR1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295527-B1 Process for the preparation of 3-aminophenyl-2-hydroxyethylsulfon BAYER AG (DE) 1994-03-02 EP disclosed
EP-0387531-B1 PROCESS FOR THE PREPARATION OF BETA-CHLOROETHYL SULFONYL ARYL ISOCYANATES HOECHST AKTIENGESELLSCHAFT (DE) 1993-05-19 EP disclosed
EP-0384265-B1 PROCESS FOR THE PREPARATION OF BETA-CHLOROETHYL SULFONYL ARYL ISOCYANATES HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-31 EP disclosed
EP-0387531-A1 Process for the preparation of beta-chloroethyl sulfonyl aryl isocyanates HOECHST AKTIENGESELLSCHAFT (DE) 1990-09-19 EP disclosed
EP-0384265-A1 Process for the preparation of beta-chloroethyl sulfonyl aryl isocyanates HOECHST AKTIENGESELLSCHAFT (DE) 1990-08-29 EP disclosed
US-4948917-A REACTING PHOSGENE AND BETA-HYDROXYETHYLSULFONYL-ARYLAMINE HOECHST AKTIENGESELLSCHAFT (DE) 1990-08-14 US disclosed
US-4929757-A Process for the preparation of 3-aminophenyl 2-hydroxy-ethyl sulphone BAYER AKTIENGESELLSCHAFT (DE) 1990-05-29 US disclosed