SCHEMBL9409098

SCHEMBL9409098

COc1cccc(Nc2cc(C(N)=O)c(C(N)=O)cc2Nc2cccc(OC)c2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.63
AKR1C2 P52895 4/20 0.63
PDE4B Q07343 3/20 0.62
SIRT2 Q8IXJ6 3/20 0.58
SIRT1 Q96EB6 1/20 0.58
NPC1 O15118 2/20 0.58
GFER P55789 2/20 0.58
GAA P10253 1/20 0.58
MTNR1A P48039 1/20 0.55
MTNR1B P49286 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.54
TP53 P04637 1/20 0.54
MAPT P10636 1/20 0.54
RAB9A P51151 1/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
POLB P06746 1/20 0.54
LMNA P02545 2/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
PARP1 P09874 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9409049 0.94 AKR1C3 (0.58) AKR1C3AKR1C2PDE4BSIRT2SIRT1
SCHEMBL28357281 0.88 SIRT2 (0.75) AKR1C3AKR1C2PDE4BSIRT2SIRT1
SCHEMBL9409067 0.83 AKR1C3 (0.60) AKR1C3AKR1C2SIRT2NPC1GFER
SCHEMBL5078980 0.83 PDE4B (0.64) AKR1C3AKR1C2PDE4BSIRT2SIRT1
SCHEMBL9409059 0.81 ALDH1A1 (0.58) AKR1C3AKR1C2SIRT2NPC1SMN1; SMN2
SCHEMBL29127204 0.81 PDE4B (0.71) AKR1C3AKR1C2PDE4BSYK
SCHEMBL30664053 0.81 PDE4B (0.71) AKR1C3AKR1C2PDE4BSYK
SCHEMBL9409184 0.80 SYK (0.57) AKR1C3AKR1C2SIRT2SIRT1GAA
SCHEMBL9594696 0.79 AKR1C3 (0.81) AKR1C3AKR1C2NPC1GFERGAA
SCHEMBL9409062 0.78 SIRT2 (0.47) PDE4BSIRT2SIRT1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0600832-A1 Derivatives of diamino benzoic and diamino phthalic acid und their use as protein linase inhibitors CIBA-GEIGY AG (CH) 1994-06-08 EP claimed
EP-0600832-A1 Derivatives of diamino benzoic and diamino phthalic acid und their use as protein linase inhibitors CIBA-GEIGY AG (CH) 1994-06-08 EP disclosed