SCHEMBL9409062

SCHEMBL9409062

COC(=O)c1cc(Nc2cccc(O)c2)c(Nc2cccc(O)c2)cc1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 7/20 0.47
BRAF P15056 4/20 0.47
MAPT P10636 1/20 0.47
ALOX15 P16050 1/20 0.47
KDR P35968 1/20 0.46
CHEK1 O14757 1/20 0.46
PAK4 O96013 1/20 0.46
CSNK2A2 P19784 1/20 0.46
CDK2 P24941 1/20 0.46
MAPK1 P28482 1/20 0.46
AKT1 P31749 1/20 0.46
MAPK8 P45983 1/20 0.46
PLK1 P53350 1/20 0.46
CSNK2B P67870 1/20 0.46
CSNK2A1 P68400 1/20 0.46
MAP2K1 Q02750 1/20 0.46
SIRT1 Q96EB6 3/20 0.45
PDE4B Q07343 2/20 0.44
PDE4A P27815 1/20 0.44
PDE4C Q08493 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9409080 0.90 BRAF (0.55) SIRT2BRAFCHEK1PAK4CSNK2A2
SCHEMBL9409034 0.86 ALDH1A1 (0.56) SIRT2MAPTALOX15MAPK1ALDH1A1
SCHEMBL9409200 0.86 AKR1C3 (0.52) SIRT2MAPTALOX15MAPK1SIRT1
SCHEMBL9409202 0.85 MAPT (0.64) SIRT2MAPTALOX15SIRT1PDE4B
SCHEMBL9409093 0.85 LMNA (0.52) SIRT2MAPTALOX15SIRT1PDE4B
SCHEMBL9409049 0.85 AKR1C3 (0.58) SIRT2MAPTSIRT1PDE4B
SCHEMBL9409026 0.84 SIRT2 (0.55) SIRT2MAPTALOX15SIRT1PDE4B
SCHEMBL9409168 0.84 AKR1C3 (0.56) SIRT2MAPTALOX15ALDH1A1
SCHEMBL9409059 0.83 ALDH1A1 (0.58) SIRT2MAPTMAPK1ALDH1A1
SCHEMBL9409066 0.82 PDE4B (0.47) SIRT2MAPTALOX15SIRT1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0600832-A1 Derivatives of diamino benzoic and diamino phthalic acid und their use as protein linase inhibitors CIBA-GEIGY AG (CH) 1994-06-08 EP disclosed