SCHEMBL9409154

SCHEMBL9409154

NC(=O)c1cc(Nc2ccc(C(=O)O)cc2)c(Nc2ccc(C(=O)O)cc2)cc1C(N)=O

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.55
AKR1C2 P52895 8/20 0.55
SIRT2 Q8IXJ6 7/20 0.51
KDM4E B2RXH2 3/20 0.50
GAA P10253 3/20 0.50
MAPT P10636 2/20 0.50
NPC1 O15118 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
GFER P55789 2/20 0.50
HSD17B10 Q99714 2/20 0.50
ALDH1A1 P00352 1/20 0.50
THRB P10828 1/20 0.50
HPGD P15428 1/20 0.50
RAB9A P51151 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9409210 0.89 SIRT2 (0.58) AKR1C3AKR1C2SIRT2KDM4EGAA
SCHEMBL2723037 0.83 SIRT2 (0.58) SIRT2KDM4EGAAMAPTGFER
SCHEMBL22725391 0.83 AKR1C3 (0.70) AKR1C3AKR1C2KDM4EGAAMAPT
SCHEMBL9409097 0.82 MAPT (0.57) AKR1C3AKR1C2SIRT2KDM4EGAA
SCHEMBL11177202 0.82 AKR1C3 (0.57) AKR1C3AKR1C2SIRT2KDM4EGAA
SCHEMBL9409036 0.81 PRKD3 (0.51) SIRT2KDM4EGAAMAPTGFER
SCHEMBL9409084 0.81 SIRT2 (0.73) AKR1C3AKR1C2SIRT2KDM4EGAA
SCHEMBL9409032 0.81 SIRT2 (0.59) AKR1C3AKR1C2SIRT2
SCHEMBL2391240 0.80 MEN1 (0.50) SIRT2MAPTALDH1A1MEN1KMT2A
SCHEMBL9409101 0.80 MAPT (0.54) AKR1C3AKR1C2SIRT2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0600832-A1 Derivatives of diamino benzoic and diamino phthalic acid und their use as protein linase inhibitors CIBA-GEIGY AG (CH) 1994-06-08 EP disclosed