SCHEMBL9414142

SCHEMBL9414142

CC(C)(C)OC(=O)NC(Cc1ccccc1)C(=O)N1CCCC1CNS(=O)(=O)CCCCN

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.51
F2 P00734 1/20 0.49
PRSS1 P07477 1/20 0.49
KMT2A Q03164 2/20 0.46
HRH2 P25021 1/20 0.45
HRH1 P35367 1/20 0.45
MAPK1 P28482 1/20 0.44
KLK5 Q9Y337 1/20 0.44
CMA1 P23946 9/20 0.44
PABPC1 P11940 1/20 0.42
CTRC Q99895 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9414140 1.00 ACE (0.51) ACEF2PRSS1KMT2AHRH2
SCHEMBL9076472 0.88 ACE2 (0.44) ACEF2PRSS1
SCHEMBL9076477 0.88 ACE2 (0.44) ACEF2PRSS1
SCHEMBL9074561 0.86 ACE2 (0.42) ACEF2PRSS1
SCHEMBL9074564 0.86 ACE2 (0.42) ACEF2PRSS1
SCHEMBL9074231 0.85 ACE (0.55) ACEF2PRSS1KMT2AHRH2
SCHEMBL9074235 0.85 ACE (0.55) ACEF2PRSS1KMT2AHRH2
SCHEMBL9073912 0.80 ACE (0.42) ACE
SCHEMBL9073915 0.80 ACE (0.42) ACE
SCHEMBL9073821 0.79 ACE2 (0.41) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623596-A1 N-acylpyrrolidines or N-acylpiperidines having a guanidinyl- or amidinyl-substituted side chain as thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-11-09 EP disclosed