SCHEMBL9418937

SCHEMBL9418937

CC(=O)c1ccc2c(c1)CC(C)(C)CC(C)(C)C2

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
MAPT P10636 2/20 0.55
HSD17B1 P14061 1/20 0.47
PGR P06401 1/20 0.41
CNR1 P21554 4/20 0.40
CNR2 P34972 4/20 0.40
HPGD P15428 1/20 0.38
KCNJ1 P48048 2/20 0.37
CYP2A6 P11509 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9419031 0.81 MAPT (0.53) NPC1RAB9AMAPTHSD17B1PGR
SCHEMBL12619017 0.78 ALDH1A1 (0.53) MAPTCNR1CNR2CA1CA2
SCHEMBL9418956 0.77 RARG (0.61) NPC1RAB9AKDM4E
SCHEMBL9418959 0.77 RARG (0.61) NPC1RAB9AKDM4E
SCHEMBL9418960 0.75 MAPT (0.55) NPC1RAB9AMAPTHSD17B1PGR
SCHEMBL17926682 0.74 MAPT (0.46) NPC1RAB9AMAPTHSD17B1PGR
SCHEMBL15927508 0.74 GSK3B (0.47) CNR1CNR2
SCHEMBL15927440 0.74 CNR1 (0.47) NPC1RAB9AMAPTCNR1CNR2
SCHEMBL21584068 0.72 NPC1 (0.67) NPC1RAB9AMAPTHSD17B1HPGD
SCHEMBL29793289 0.72 NPC1 (0.67) NPC1RAB9AMAPTHSD17B1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP disclosed
US-4992574-A Skin disorders, antiallergens, antiinflammatory agent HOFFMANN-LA ROCHE INC. (US) 1991-02-12 US disclosed
EP-0315071-A2 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed