SCHEMBL9419059

SCHEMBL9419059

CC(=O)c1ccc2c(c1)CCC(C)CC2

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
MAPT P10636 3/20 0.55
HSD17B1 P14061 1/20 0.47
ALDH1A1 P00352 3/20 0.46
HPGD P15428 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
KCNJ1 P48048 1/20 0.42
SMYD3 Q9H7B4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12778355 0.90 NPC1 (0.51) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL29793289 0.85 NPC1 (0.67) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL21584068 0.85 NPC1 (0.67) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL1466022 0.81 NPC1 (0.67) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL31048932 0.81 NPC1 (0.67) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL33121 0.81 ALDH1A1 (0.68) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL22627409 0.79 NPC1 (0.65) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL9419020 0.79 NPC1 (0.65) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL9143187 0.79 MAPT (0.44) NPC1RAB9AMAPTHSD17B1ALDH1A1
SCHEMBL19231579 0.78 NPC1 (0.58) NPC1RAB9AMAPTHSD17B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP disclosed
US-4992574-A Skin disorders, antiallergens, antiinflammatory agent HOFFMANN-LA ROCHE INC. (US) 1991-02-12 US disclosed
EP-0315071-A2 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed