SCHEMBL9419641

SCHEMBL9419641

O=C(CN1CCCCC1)N1c2ccccc2Oc2ccccc21

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.62
ALOX15 P16050 2/20 0.62
USP2 O75604 2/20 0.62
P2RX4 Q99571 4/20 0.61
GAA P10253 2/20 0.52
MAPT P10636 1/20 0.52
CACNA1H O95180 1/20 0.51
CACNA1B Q00975 1/20 0.51
POLB P06746 2/20 0.50
RAD52 P43351 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 1/20 0.49
KDM4E B2RXH2 1/20 0.47
PKM P14618 1/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9419617 0.98 ALDH1A1 (0.64) ALDH1A1ALOX15USP2P2RX4GAA
SCHEMBL6045372 0.89 USP2 (0.51) ALDH1A1ALOX15USP2P2RX4TP53
SCHEMBL6045322 0.87 USP2 (0.52) ALDH1A1ALOX15USP2P2RX4TP53
SCHEMBL9419650 0.87 HTT (0.54) ALDH1A1ALOX15USP2P2RX4GAA
SCHEMBL5453524 0.82 P2RX4 (0.50) ALDH1A1ALOX15USP2P2RX4MEN1
SCHEMBL6045315 0.77 MEN1 (0.53) ALDH1A1P2RX4GAAMAPTMEN1
SCHEMBL5242431 0.74 ALDH1A1 (0.44) ALDH1A1ALOX15USP2P2RX4KDM4E
SCHEMBL5241094 0.74 P2RX4 (0.65) P2RX4
SCHEMBL5451618 0.73 LTA4H (0.48) ALDH1A1GAAPKMTP53
SCHEMBL5460660 0.73 TP53 (0.43) ALDH1A1ALOX15USP2P2RX4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371081-A Useful in potentiating the cytotoxic effect of chemotherapeutic agents ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 1994-12-06 US claimed
WO-1993003729-A1 N-SUBSTITUTED PHENOXAZINES FOR TREATING MULTIDRUG RESISTANT CANCER CELLS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1993-03-04 WO claimed
US-5371081-A Useful in potentiating the cytotoxic effect of chemotherapeutic agents ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 1994-12-06 US disclosed
WO-1993003729-A1 N-SUBSTITUTED PHENOXAZINES FOR TREATING MULTIDRUG RESISTANT CANCER CELLS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1993-03-04 WO disclosed