SCHEMBL9425879

SCHEMBL9425879

CC(C)(C)OC(=O)N[C@@H](CO)C(=O)NCCCCC1CCCCC1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.57
CTSK P43235 4/20 0.57
NMT1 P30419 6/20 0.49
NMT2 O60551 5/20 0.49
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CAPN1 P07384 1/20 0.46
BCHE P06276 1/20 0.45
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
EPHX1 P07099 1/20 0.41
CACNA1B Q00975 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9718268 0.91 CTSS (0.60) CTSSCTSKNMT1NMT2HDAC4
SCHEMBL9425883 0.83 CTSS (0.45) CTSSCTSKNMT1NMT2HDAC4
SCHEMBL1861303 0.81 CTSK (0.69) CTSSCTSKNMT1NMT2HDAC4
SCHEMBL1861306 0.81 CTSK (0.69) CTSSCTSKNMT1NMT2HDAC4
SCHEMBL506749 0.80 CTSK (0.55) CTSSCTSKCAPN1TDP1EPHX1
SCHEMBL21561570 0.80 CTSK (0.55) CTSSCTSKCAPN1TDP1EPHX1
SCHEMBL506750 0.80 CTSK (0.55) CTSSCTSKCAPN1TDP1EPHX1
SCHEMBL5967594 0.78 CTSS (0.52) CTSSCTSKCAPN1TDP1
SCHEMBL12143788 0.78 CTSS (0.52) CTSSCTSKCAPN1TDP1
SCHEMBL4073139 0.78 EPHX1 (0.60) CTSSCTSKKMT2ATDP1EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5290799-A 7-oxabicycloheptyl substituted heterocyclic thioamide prostaglandin analogs useful in the treatment of thrombotic and vasospastic disease E. R. SQUIBB & SONS, INC. (US) 1994-03-01 US disclosed
EP-0544287-A1 Gem-dialkyl-7-oxabicycloheptyl substituted heterocyclic amide prostaglandin analogs useful in the treatment of thrombotic and vasospastic disease E.R. SQUIBB & SONS, INC. (US) 1993-06-02 EP disclosed
US-5153327-A 7-Oxabicycloheptyl substituted heterocyclic amide or ester prostaglandin analogs useful in the treatment of thrombotic and vasospastic disease E. R. SQUIBB & SONS, INC. (US) 1992-10-06 US disclosed
US-5100889-A Thromboxane A2 receptor antagonists, thromboxane synthetase inhibitor E. R. SQUIBB & SONS, INC. (US) 1992-03-31 US disclosed