SCHEMBL94267

SCHEMBL94267

CC(=O)c1cccc2nc3ccccc3nc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.70
MAPT P10636 8/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
KMT2A Q03164 5/20 0.52
RAB9A P51151 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
GAA P10253 2/20 0.52
HTT P42858 2/20 0.49
THRB P10828 1/20 0.49
MEN1 O00255 3/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
NQO2 P16083 1/20 0.47
NPC1 O15118 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
KDM4E B2RXH2 3/20 0.45
ATM Q13315 1/20 0.45
PABPC1 P11940 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL123790 0.90 ALDH1A1 (0.63) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
Maleic Acid SCHEMBL1155758 0.90 ALDH1A1 (0.63) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL19971558 0.87 ALDH1A1 (0.73) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL28382224 0.84 ALDH1A1 (0.75) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL31598603 0.84 ALDH1A1 (0.50) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
Phenazine-1-Carboxylic Acid SCHEMBL27752237 0.83 ALDH1A1 (0.93) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL26523348 0.83 ALDH1A1 (0.49) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
Phenazine-1-Carboxylic Acid SCHEMBL29370801 0.82 ALDH1A1 (1.00) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
Phenazine-1-Carboxylic Acid SCHEMBL122864 0.82 ALDH1A1 (1.00) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19
Phenazine-1-Carboxylic Acid SCHEMBL28160016 0.82 ALDH1A1 (1.00) ALDH1A1MAPTCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5425 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106917-A1 EDIBLE TRANSMUCOSAL DRUG DELIVERY METHOD USING AN INTERMEDIATE CAPSULE AS A TEMPORARY VESSEL BioPhysics Pharma, Inc. (US) 2026-05-21 WO claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
EP-4654963-A1 TREATMENT OF MENTAL ILLNESS VIA ADMINISTRATION OF BUNTANETAP AND ANALOGUES THEREOF Annovis Bio, Inc. (US) 2025-12-03 EP claimed
EP-4618973-A1 METHODS OF SWITCHING NEUROPSYCHIATRIC MEDICATIONS USING ULOTARONT Sumitomo Pharma America, Inc. (US) 2025-09-24 EP claimed
US-20250268841-A1 Trans-Epithelial Membrane Drug Delivery System Masiz, John J. (US) 2025-08-28 US claimed
US-20250191770-A1 COMPUTERIZED DECISION SUPPORT TOOL AND MEDICAL DEVICE FOR RESPIRATORY CONDITION MONITORING AND CARE PFIZER INC. (US) 2025-06-12 US claimed
US-20250179064-A1 BENZOQUINOLONE INHIBITORS OF VMAT2 AUSPEX PHARMACEUTICALS LLC 2025-06-05 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-3334725-B1 BROMODOMAIN AND EXTRA TERMINAL (BET) INHIBITOR AND A PROTEIN PHOSPHATASE 2A (PP2A) ACTIVATOR FOR TREATING BET INHIBITOR RESISTANT CANCER DANA FARBER CANCER INST INC (US) 2025-04-23 EP claimed
US-20250120907-A1 Transmucosal Drug Delivery System Masiz, John J. (US) 2025-04-17 US claimed
US-4996047-A Sustained release drug-resin complexes RICHARDSON-VICKS, INC. (US) 1991-02-26 US claimed
EP-0367746-A2 Sustained release drug-resin complexes RICHARDSON-VICKS, INC. (US) 1990-05-09 EP claimed
EP-0174342-B1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1989-12-20 EP claimed
EP-0222425-A2 Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1987-05-20 EP claimed
EP-0218300-A2 Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1987-04-15 EP claimed
EP-0174342-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES. UNIV FLORIDA (US) 1986-03-19 EP claimed
WO-1985003937-A1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1985-09-12 WO claimed
EP-0110955-A1 BRAIN-SPECIFIC DRUG DELIVERY. UNIV FLORIDA (US) 1984-06-20 EP claimed
WO-1983003968-A1 BRAIN-SPECIFIC DRUG DELIVERY UNIVERSITY OF FLORIDA (US) 1983-11-24 WO claimed
US-4175119-A Composition and method to prevent accidental and intentional overdosage with psychoactive drugs PORTER GARRY L 1979-11-20 US claimed