SCHEMBL9426795

SCHEMBL9426795

CS(=O)(=O)Nc1ccc(Sc2cnc(N)s2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 1/20 0.42
HPGD P15428 2/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
LIMK1 P53667 2/20 0.39
PRKD3 O94806 2/20 0.39
ROCK1 Q13464 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
CHEK1 O14757 1/20 0.39
CDK8 P49336 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
CDC7 O00311 1/20 0.39
PLK4 O00444 1/20 0.39
DAPK3 O43293 1/20 0.39
DYRK3 O43781 1/20 0.39
JAK2 O60674 1/20 0.39
ROCK2 O75116 1/20 0.39
MAP4K4 O95819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9426024 0.79 CCNE1 (0.47) HPGDCDK1CDK2ALDH1A1PIP4K2A
SCHEMBL9426820 0.78 GAA (0.42) CA12CA1CA2CA9CDK2
SCHEMBL5171580 0.75 CYP3A4 (0.48) PLK4CDK2ALDH1A1MYCWDR5
SCHEMBL28014672 0.75 PTGIR (0.58) PTGIRHPGDCA12CA1CA2
SCHEMBL9048249 0.74 NOS1 (0.46) HPGDLIMK1CDK2KDM4EALDH1A1
SCHEMBL9426129 0.72 NR1H2 (0.45) CDK2CSNK2A1ALDH1A1HTTMYC
SCHEMBL15587224 0.72 MYC (0.47) HPGDCDK2CSNK2A1ALDH1A1LMNA
SCHEMBL9426921 0.72 POLB (0.51) PTGIRHPGDKDM4EALDH1A1LMNA
SCHEMBL9426995 0.70 CA12 (0.42) HPGDCA12CA1CA2CA9
SCHEMBL1060492 0.70 MAPT (0.54) HPGDKDM4EALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1027370-C Process for preparing thiazole derivatives FUJISAWA FARMACEUTICAL CO LTD (JP) 1995-01-11 CN disclosed
US-5369107-A Thiazole derivatives, processes for production thereof and pharmaceutical compositions comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-11-29 US disclosed
US-5256675-A Antirheumatic agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-10-26 US disclosed
CN-1049337-A Thiazole derivative prepares their method, and the medicinal compositions that contains them FUJISAWA PHARMACEUTICAL CO (JP) 1991-02-20 CN disclosed
EP-0412404-A2 Thiazole derivatives, processes for production thereof and pharmaceutical compositions comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-02-13 EP disclosed