SCHEMBL9428013

SCHEMBL9428013

Cn1c(N2CCN(CCCOc3ccc(C(=O)c4ccccc4)cc3NS(C)(=O)=O)CC2)cc(=O)n(C)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 13/20 0.46
HRH3 Q9Y5N1 2/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.42
ADRA1A P35348 3/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1B P35368 2/20 0.41
HRH4 Q9H3N8 1/20 0.41
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
HRH2 P25021 1/20 0.40
LMNA P02545 1/20 0.40
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
CYP3A4 P08684 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9429177 0.99 HRH1 (0.45) HRH1HRH3KDM4EALDH1A1ADRA1A
SCHEMBL9428145 0.86 HRH1 (0.45) HRH1HRH3ADRA1AADRA1DADRA1B
SCHEMBL9428617 0.86 HRH1 (0.48) HRH1ALDH1A1ADRA1AADRA1DADRA1B
Hydrochloric Acid SCHEMBL9428851 0.85 MAPT (0.49) HRH1ALDH1A1ADRA1AADRA1DADRA1B
Oxalic Acid SCHEMBL9428453 0.85 HRH1 (0.44) HRH1KDM4EALDH1A1ADRA1AADRA1D
SCHEMBL9428524 0.84 HRH1 (0.49) HRH1HRH3KDM4EALDH1A1ADRA1A
SCHEMBL9428782 0.84 HRH1 (0.49) HRH1HRH3KDM4EALDH1A1ADRA1A
Hydrochloric Acid SCHEMBL9428272 0.83 MAPT (0.41) HRH1HRH3KDM4EALDH1A1ADRA1A
SCHEMBL9428899 0.82 ADRA1B (0.40) HRH1ALDH1A1ADRA1AADRA1DADRA1B
SCHEMBL9384791 0.81 KDM4E (0.48) HRH1HRH3KDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed