SCHEMBL9431007

SCHEMBL9431007

CN(N=O)C(=O)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MITF O75030 1/20 0.45
FFAR1 O14842 1/20 0.44
TSHR P16473 1/20 0.43
CA2 P00918 3/20 0.43
CA12 O43570 2/20 0.43
CA9 Q16790 2/20 0.43
CA1 P00915 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
PTPN11 Q06124 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691754 0.85 ALDH1A1 (0.50) ALDH1A1MEN1KMT2ATSHRCA2
SCHEMBL8934937 0.82 TSHR (0.63) EPHX2NR1H4ALDH1A1PKMMEN1
Hydrochloric Acid SCHEMBL28761138 0.81 ALDH1A1 (0.50) NR1H4ALDH1A1MEN1KMT2ATSHR
SCHEMBL10968223 0.76 TSHR (0.50) ALDH1A1MEN1KMT2ATSHRCA2
SCHEMBL5445025 0.72 HTT (0.51) EPHX2NR1H4ALDH1A1PKMMEN1
Acedoben SCHEMBL24320 0.71 ALDH1A1 (0.68) EPHX2NR1H4ALDH1A1MEN1KMT2A
SCHEMBL4745756 0.71 EPHX2 (0.71) EPHX2NR1H4ALDH1A1MEN1KMT2A
SCHEMBL9555249 0.71 ALDH1A1 (0.61) EPHX2NR1H4ALDH1A1PKMMEN1
SCHEMBL1066727 0.70 MAPT (0.59) ALDH1A1CA2CA12CA9CA1
Hydrochloric Acid SCHEMBL7563130 0.70 EPHX2 (0.47) EPHX2NR1H4ALDH1A1PKMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5310752-A Distamycin A analogs; antitumor agents, viricides FARMITALIA CARLO ERBA SPA (IT) 1994-05-10 US disclosed
EP-0246868-B1 SITE SPECIFIC ALKYLATING AGENTS FARMITALIA CARLO ERBA S.r.l. (IT) 1992-09-16 EP disclosed
US-5017599-A Antitumor, antiviral distamycin A analog FARMITALIA CARLO ERBA, SPA (IT) 1991-05-21 US disclosed
EP-0246868-A1 Site specific alkylating agents FARMITALIA CARLO ERBA S.r.l. (IT) 1987-11-25 EP disclosed