SCHEMBL8934937

SCHEMBL8934937

CN(C)C(=O)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.63
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
APEX1 P27695 1/20 0.53
ALDH1A1 P00352 1/20 0.52
EPHX2 P34913 1/20 0.51
NR1H4 Q96RI1 1/20 0.51
PKM P14618 1/20 0.50
MITF O75030 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
FFAR1 O14842 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687878 0.87 TSHR (0.79) TSHRCA12CA1CA2CA9
SCHEMBL11713193 0.83 ALDH1A1 (0.66) TSHRALDH1A1MEN1KMT2AFFAR1
SCHEMBL3649965 0.82 TSHR (0.61) TSHRCA12CA1CA2CA9
SCHEMBL9431007 0.82 EPHX2 (0.46) TSHRCA12CA1CA2CA9
Fenuron SCHEMBL9451054 0.81 TSHR (0.64) TSHRCA12CA1CA2CA9
Fenuron SCHEMBL62004 0.81 TSHR (0.64) TSHRCA12CA1CA2CA9
Fenuron SCHEMBL8366971 0.81 TSHR (0.64) TSHRCA12CA1CA2CA9
Fenuron SCHEMBL10806698 0.81 TSHR (0.64) TSHRCA12CA1CA2CA9
SCHEMBL8887134 0.81 MEN1 (0.64) TSHRALDH1A1MEN1KMT2A
SCHEMBL7821470 0.80 SLC1A3 (0.47) TSHRAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996030329-A1 SUBSTITUTED BENZENE DERIVATIVES USEFUL AS NEURAMINIDASE INHIBITORS BIOCRYST PHARMACEUTICALS, INCORPORATED (US) 1996-10-03 WO disclosed